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1-(5-chloropyridin-2-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-(2-fluoro-4-methoxyphenyl)-5-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
1-methyl-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazine-2-carboxylic acid
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-N-ethyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1R,2S)-N-butyl-2-[3-(4-fluorophenoxy)azetidine-1-carbonyl]cyclohexane-1-carboxamide
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
2-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-decahydroisoquinoline
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-5-carboxamide
4-[1-(2,1,3-benzothiadiazol-5-ylmethyl)-1H-imidazol-2-yl]-2-methoxyphenol
4-(4-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
methyl 4-(5-methyl-4-{[methyl({[4-(trifluoromethyl)phenyl]methyl})amino]methyl}-1,3-oxazol-2-yl)benzoate
8-(2,6-dimethoxybenzoyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-3-(1,2-oxazolidin-2-yl)propan-1-one
(1-ethyl-5-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
3-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
5-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
4-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-fluoro-N,3-dimethyl-N-[2-(phenylsulfanyl)ethyl]-1H-indole-2-carboxamide
N-{2-methyl-1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}methanesulfonamide
4-{1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}benzoic acid
1-[2-(3-cyclopentylpropanamido)ethyl]-N-phenyl-1H-1,2,3-triazole-4-carboxamide
methyl 1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
4-(2-methyl-1,3-benzoxazole-6-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-methyl-N-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}benzene-1-sulfonamide
1-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
(4S)-1-[4-(difluoromethoxy)benzoyl]-3,3,4-trimethylpiperidin-4-ol
2-methoxy-N-({3-methyl-7-[3-(prop-2-en-1-yloxy)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-phenylacetamide
1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-[(3-methylpyridin-2-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
(3S,9aR)-3-(cyclohexylmethyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[6-(methoxymethyl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N,2-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
2-[1-(1H-1,2,3-benzotriazol-5-yl)-1H-imidazol-2-yl]quinoline
7-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1-benzofuran-2-carboxamide
N,N-bis(propan-2-yl)-2-(pyrimidin-2-yl)benzamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(1-benzylpyrrolidin-3-yl)methyl]-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
2-methyl-9-[(4-methylthiophen-2-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(1R,5R)-6-[(3-cyanophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(dimethylamino)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}pyridine
1-(4-methoxybenzoyl)-4-(1-methylpiperidine-2-carbonyl)piperazine
6-(2-aminoethyl)-N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methylpyrimidin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-chloro-5-acetamido-N-methylbenzamide