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3-[(3,4-difluorophenyl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-[3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
(benzylsulfamoyl)[1-(pyrazin-2-yl)propan-2-yl]amine
2-(4-methyl-1,4-diazepan-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]acetamide
2-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-benzofuran-5-carboxamide
2-methoxy-6-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(2-hydroxy-2-methylpropanoyl)piperidin-4-yl]propanamide
[(1R,3S,3aS,6aR)-1,5-dimethyl-3-[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-oxoethyl)urea
N4-methyl-6-(4-methylpiperazin-1-yl)-N4-(quinolin-4-ylmethyl)pyrimidine-2,4-diamine
2-ethyl-1-(9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.5]undecan-3-yl)butan-1-one
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-2,3-dihydro-1H-indene-1-carboxamide
7-[1-(2-fluoroethyl)-4-phenyl-1H-imidazol-5-yl]-4-methyl-2H-chromen-2-one
N-({7-[3-(furan-2-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
N-ethyl-1-(2-methylpropyl)-5-oxo-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-{5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
6-cyano-N-ethyl-N-[(2-fluorophenyl)methyl]pyridine-3-carboxamide
3-ethyl-5-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazole-4-carboxamide
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[(5-oxo-1-propylpyrrolidin-3-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)morpholine
3-(2-methyl-1H-indol-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]propanamide
N-(oxolan-2-ylmethyl)-3-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]propanamide
1-(difluoromethyl)-N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
6-methoxy-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-(3-chloro-4-methoxyphenyl)-3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]propanamide
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
2,5-dimethyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-{1H-pyrrolo[2,3-b]pyridin-6-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-[3-(cyclopropylmethyl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl]pyridine
{4-[(4-methoxyphenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}methanol
2-(5-fluoro-2-methylphenyl)-2-(4-{[(propan-2-yl)carbamoyl]methyl}piperazin-1-yl)acetic acid
3-[1-(5-fluoropyridin-2-yl)-1H-pyrazol-4-yl]propanoic acid
N1,N1,N3-trimethyl-N3-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-1,3-dicarboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
3-{2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
3-{[(1-hydroxycyclohexyl)methyl]sulfamoyl}-N-[2-(methylamino)ethyl]benzamide
2-amino-4-(3-chloro-4-hydroxyphenyl)-6-(2-methylpropanoyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
7-cyclohexyl-2-cyclopentanecarbonyl-2,7-diazaspiro[4.5]decan-6-one
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
5-[(4-methoxyphenyl)methyl]-5-(3-oxo-3-{spiro[indene-1,4'-piperidine]-1'-yl}propyl)pyrrolidin-2-one
N-[1-(2-fluorophenyl)piperidin-4-yl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
N-ethyl-2-{4-[5-(methoxymethyl)thiophene-2-carbonyl]piperazin-1-yl}acetamide
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-ethyl-1-[(5-methylfuran-2-yl)methyl]urea