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N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(pyridine-3-carbonyl)piperidine-4-carboxamide
2-(2-methoxyethyl)-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(1H-pyrazol-1-yl)butanamide
1-{5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperidine-3-carboxamide
2-butyl-8-(3-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[2-({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]benzene-1-sulfonamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,6-dimethylpyrimidine-4-carboxamide
N-ethyl-5-(2-methoxyphenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
2-{imidazo[1,2-a]pyridin-3-yl}-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
N,7-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-amino-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-phenylpyrimidine-5-carboxamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(1H-indazol-1-yl)propyl]propanamide
3-methyl-1-propyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-pyrazole-4-carboxamide
3-({[1-ethyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
2-methyl-6-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}pyrimidin-4-amine
6-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
1-(furan-2-carbonyl)-4-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperazine
1-(2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(propylsulfanyl)ethyl]pyrimidine-5-carboxamide
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(dimethylamino)ethyl]acetamide
6-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2,4-dimethylpyridine-3-carbonitrile
5-{2,7-diazaspiro[4.5]decane-7-carbonyl}-N-phenylpyrimidin-2-amine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
2-(2,4,6-trimethylphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}-N,N-dimethylpyrazine-2-carboxamide
2-[3-({[1-(cyclohexylmethyl)piperidin-3-yl]amino}methyl)phenoxy]ethan-1-ol
N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(cyclobutylmethyl)-2-(isoquinolin-5-ylmethyl)-2,7-diazaspiro[4.5]decane
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}furan-3-carboxamide
2-{4-[4-(2-fluorophenoxy)piperidin-1-yl]piperidin-1-yl}-7-methanesulfonyl-4-methylquinazoline
1-cyclobutanecarbonyl-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]piperidine-4-carboxamide
1-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-{7-[4-(methylsulfanyl)benzoyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
N-ethyl-1,3-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-({3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-2-methyl-1,3-benzothiazole
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
dimethyl(2-{2-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
(3S,4R)-1-[4-(diethylamino)benzoyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
(3aS,7aR)-5-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
methyl 3-[(5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]propanoate
(4aS,8aR)-6-[(4-methylpiperazin-1-yl)sulfonyl]-1-propyl-decahydro-1,6-naphthyridin-2-one