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2-oxo-N-(thiophen-3-ylmethyl)-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-[(prop-2-en-1-yl)amino]-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}benzamide
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
(4-{[1-(isoquinoline-1-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-2-(4-phenyl-1H-imidazol-1-yl)acetamide
(2S,4S)-4-amino-N-methyl-1-{[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]sulfonyl}pyrrolidine-2-carboxamide
4-{[(2,2-dimethyloxan-4-yl)(ethyl)amino]methyl}-6,8-dimethyl-2H-chromen-2-one
4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-(3,4-dimethylphenyl)-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidin-3-amine
8-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4,4,4-trifluoro-3-{3-[(4-fluorophenyl)formamido]propanamido}butanoic acid
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(2-hydroxyethyl)-5-[2-(2-methyl-1H-indol-3-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-2-(5-methyl-1H-pyrazol-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
2-butyl-N-(2-fluoro-5-propanamidophenyl)-2,5-dihydro-1H-pyrrole-1-carboxamide
(2R,6R)-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-{5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
4-[5-(3-benzyl-1H-1,2,4-triazol-5-yl)furan-2-yl]-2-methylbut-3-yn-2-ol
4-{[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
(3S,4R)-4-(3-methoxyphenyl)-1-sulfamoylpyrrolidine-3-carboxylic acid
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[2-(1H-indol-3-yl)ethyl]amino}acetamide
6-{4-[1-(dimethylamino)ethyl]phenyl}-N-methylpyridazin-3-amine
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
4-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-(1H-indazol-6-yl)piperazin-2-one
3-(3-fluorophenyl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-pyrazole-4-carboxamide
N,N-diethyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
4-{5-[(1S,3R)-3-aminocyclopentyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
N-[4-(3-fluorophenyl)phenyl]-1-(pyrimidin-2-ylmethyl)piperidine-3-carboxamide
(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
3-fluoro-6-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-(oxolan-3-yl)-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazole
3-amino-1-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}pyrrolidine-3-carboxylic acid
(3S,5R)-N3-(4-methylphenyl)-N5-[(6-methylpyridin-2-yl)methyl]piperidine-3,5-dicarboxamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-methyl-2,3-dihydro-1H-indole
1-{4-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
2-(4-methylpentyl)-4-[4-(4-methylpiperazin-1-yl)benzoyl]morpholine
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
(3R,4R)-4-amino-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-3-ol
3-(propan-2-yl)-5-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
[(3R,4R)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-amino-7-[2-(pyridin-4-ylsulfanyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(dimethyl-1,3-thiazol-5-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}dimethylamine
4-(2-methoxyphenoxy)-1-(2-methylfuran-3-carbonyl)piperidine
1-(2-methoxyethyl)-3-methyl-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione