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(2S,4R)-1-(2,2-diphenylethyl)-4-[(1-ethylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{2-methyl-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}imidazolidin-2-one
2-(2,2-dimethyloxan-4-yl)-4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}propanamide
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)acetamide
3-{cyclopropyl[(2-ethoxyphenyl)methyl]amino}propane-1,2-diol
3-(4-chlorophenyl)-5-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-1,2,4-oxadiazole
2-ethyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[2-(dimethylamino)ethyl]-3-({1-[(2R)-2-hydroxypropanoyl]piperidin-4-yl}oxy)-4-methoxybenzamide
2-(5-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}furan-2-yl)benzonitrile
2-[(3-methoxyphenyl)methyl]-8-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}propane-1-sulfonamide
1-(2-aminoethyl)-N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-(4-chlorophenyl)-N-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
2-methyl-6-[3-(propan-2-yl)-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl]pyridine
1-[(3-chloro-5-fluorophenyl)methyl]-3-(2-methoxyphenoxy)azetidine
5-methyl-N-{4-[2-(2-methyl-1H-imidazol-1-yl)propanamido]phenyl}furan-2-carboxamide
(1S,5R)-3-(1,4-dithiepan-6-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methylfuran-3-carboxamide
ethyl 4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
6-(methoxymethyl)-1-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(dimethylamino)-N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-(4-fluorophenyl)acetamide
2-{4-[(5-ethylfuran-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-cyclopropyl-1-[1-(2-hydroxybenzoyl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-2-{[(3-fluoro-4-methoxyphenyl)methyl]amino}-3-phenylpropanamide
2-amino-6-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-({[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-3,5-dimethylpyridin-4-ol
2-amino-6-(2,2-dimethyloxan-4-yl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5-methylpyridine-3-carbonitrile
N-methyl-N-[1-(pyridin-3-yl)pentyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-ethyl-4-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyridine-3-carboxamide
methyl 2-(3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamido)acetate
2-(2-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
N-{[1-(pyridine-3-sulfonyl)piperidin-3-yl]methyl}furan-2-carboxamide
9-[3-(4-hydroxyphenyl)propanoyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-1-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)cyclobutanecarboxamide
N6-(1H-indol-4-ylmethyl)-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(2S,4S)-4-amino-1-[3-(1H-imidazol-2-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
N-(2-methoxyethyl)-3,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
1-ethyl-N-[(3-fluorophenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-oxo-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
2-methyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane