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1-[(2E)-2-methylbut-2-en-1-yl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
(3S,4S)-1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidine-3,4-diol
4'-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-({1-[6-(pyridin-3-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
2-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
2-[3-(furan-2-yl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-{2-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-2-(1H-pyrazol-1-yl)butanamide
3-[(3S)-1-benzylpiperidin-3-yl]-1-(6-methoxypyridin-3-yl)urea
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(pyridin-3-yl)piperazine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
5-methyl-1-propyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-(1'-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
2-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
(4aR,7aS)-1-(3-methylbutanoyl)-4-(thiophen-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
4-(4-methanesulfonylphenyl)isoquinoline
N-{[1-(1H-imidazol-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-3-methoxybenzamide
N-[2-(3-methylpyridin-2-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3,5-dimethoxy-2-{[2-(methylcarbamoyl)piperidin-1-yl]methyl}benzoic acid
(2S,4S)-N-ethyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(furan-3-amido)pyrrolidine-2-carboxamide
N-({1-[(5-ethylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
(4aS,7aR)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}phenol
N-(2-hydroxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
(4aR,7aS)-1-{2-[4-(propan-2-yl)piperazin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(3-fluorophenyl)ethyl]-5-[4-(3-methoxypropyl)piperidine-1-carbonyl]piperidin-2-one
N-{[2-(1H-imidazol-2-yl)phenyl]methyl}-N,1-dimethylpyrrolidin-3-amine
N-(2-{[2-(cyclopropylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)acetamide
5-chloro-6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-3-carboxylic acid
4-[(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-2-yl)methyl]morpholine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
1-(2-aminoethyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoxaline
1-cyclopentyl-5-(1-methyl-1H-1,2,4-triazol-5-yl)piperidin-2-one
1-{3-[2-(furan-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
7-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-3,5-bis(trifluoromethyl)benzamide
N-(2-hydroxyethyl)-2,8-dimethyl-N-[(5-methylthiophen-2-yl)methyl]quinoline-4-carboxamide
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-(4-phenylpiperidin-1-yl)ethan-1-one
2-(3,5-difluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-(2,6-difluoro-3-methoxybenzoyl)-3-(2-ethylphenoxy)azetidine
4-[1-(propylcarbamoyl)piperidin-3-yl]benzoic acid
(2,1,3-benzothiadiazol-5-ylmethyl)({[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl})methylamine
4-ethyl-1-[2-(4-fluorophenoxy)ethyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-hydroxy-1-phenylethyl)-5-(4-methoxyphenyl)furan-2-carboxamide