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N-[(2R,4S,6R)-2-(4-chlorophenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]oxan-4-yl]acetamide
5-[1-(2,6-dimethylhept-5-en-1-yl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(ethoxymethyl)pyrimidine
N-(piperidin-3-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
3-(1H-pyrazol-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]benzamide
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
6-[(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)amino]pyridine-3-carbonitrile
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]acetic acid
4-{10-azabicyclo[4.3.1]decane-10-carbonyl}-7-methyl-2-(pyrimidin-5-yl)quinoline
N-benzyl-1-(2-{[3-(dimethylamino)phenyl]formamido}ethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-methyl-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3R,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
4-ethyl-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-cyclobutyl-6-methyl-2-(3-phenylpiperazin-1-yl)pyrimidine
3-(1,3-dihydro-2-benzofuran-5-yl)-1-[1-(2,5-dimethoxyphenyl)ethyl]urea
4-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
ethyl 2-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-2-yl}acetate
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
(2S)-2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-3-phenylpropanamide
5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
N-[(5-methylpyrazin-2-yl)methyl]-3-phenyladamantane-1-carboxamide
8-(3-chlorothiophene-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
4-{3-methylimidazo[1,5-a]pyridin-1-yl}-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-({6-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]quinazolin-4-yl}amino)ethan-1-ol
N-cyclopropyl-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
N-cyclopropyl-1-{1-[2-(1H-imidazol-1-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyridine-3-carboxamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanoyl]piperazin-2-one
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-{1-[2-(2,4,6-trifluorophenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
13-(3-phenyl-1,2,4-oxadiazol-5-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
4-chloro-3-{[(oxan-4-ylmethyl)carbamoyl]amino}-N-propylbenzamide
3-cyclohexyl-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-1H-pyrazole-4-carboxamide
(2R)-3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propane-1,2-diol
3-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}-N-(3,5-dimethylphenyl)propanamide
3-[5-(3-propyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-{4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
(2S,5R)-1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-cyclopentyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]pyrrolidin-3-yl]acetamide
N3-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-cyclopentyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2,3-dimethyl-6-[2-(morpholin-3-yl)acetyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(3-fluorophenoxymethyl)-1,3-oxazole
(2S)-2-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}-2-phenylethan-1-ol