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2-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline
2-(2-{[(2-methoxyphenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(4aS,7aR)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3R,4S)-4-(morpholin-4-yl)-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-yl]propan-1-ol
1'-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(5-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
1-[2-(1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
3-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
[(3S,5R)-1-(4-chlorobenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
{4-[(2-chlorophenyl)methyl]-1-(3-phenylprop-2-yn-1-yl)piperidin-4-yl}methanol
3-[(3R,4S)-1-[2-(4-fluorophenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(4-hydroxyphenyl)methyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
1-{3,5-dimethyl-4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
methyl 3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]benzoate
4-[(2S)-2-amino-3-cyclohexylpropanoyl]-1-(2-methoxyphenyl)piperazin-2-one
N,2,2-trimethyl-N-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}oxan-4-amine
3-{[(2-chlorophenyl)formamido]methyl}-N-ethylpiperidine-1-carboxamide
[(3S,7S)-5-(2-methyl-1,3-thiazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]propanamide
N-(2,3-dimethylquinoxalin-6-yl)-4-(pyridin-3-yl)piperazine-1-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}propan-1-one
3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)-1,3-oxazolidin-2-one
5-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[2-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-[(4-methylphenyl)methyl]-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
4-methoxy-2-[(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
propan-2-yl 4-chloro-3-[(2S,4R)-4-hydroxypyrrolidine-2-amido]benzoate
2-(4-{[methyl(2-phenoxyethyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-one
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-(2-phenylphenyl)piperazin-2-one
1-(3-chlorophenyl)-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenyl-1H-pyrazole-4-carboxamide
N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
3-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2,7-trimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
8-(3-acetyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(2-chloro-6-methoxyphenyl)-2-methylphenoxy]acetamide
{1-[(3-methylpyridin-2-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
4-[7-(5-chloropyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
2-{[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]oxy}pyrimidine
(5S)-5-{[benzyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]methyl}pyrrolidin-2-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(5-methylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6-(2-aminoethyl)-N-[(2-methoxyphenyl)methyl]-2-methylpyrimidin-4-amine
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one