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2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(3S,4R)-1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(4aS,7aR)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]ethyl}morpholine
2-{4-[(2,2-dimethylpiperazin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
N-[(1-methylpiperidin-4-yl)methyl]-4-(2-methylpropyl)benzamide
1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
6-methyl-4-oxo-2-(2-phenylethyl)-N-(propan-2-yl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[N-methyl-1-(2,6,8-trimethylquinolin-4-yl)formamido]-2-(pyridin-3-yl)acetic acid
N2-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
2-{[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one
N,N-dimethyl-5-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]pyridin-2-amine
(1R,2S,9R)-11-(5-methylpyrazine-2-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2,4-dimethyl-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}pyrimidine
5-cyclopropanecarbonyl-1'-(4-methyl-1H-imidazole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(2-methoxyethyl)-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
6-methoxy-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-1,3-benzothiazol-2-amine
1-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
(4aR,7aS)-1-pentanoyl-4-[3-(1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
2-(1H-1,3-benzodiazol-1-yl)-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]propan-1-one
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(3-hydroxypropyl)-1,4-diazepan-6-ol
(2S,4S)-4-acetamido-N-ethyl-1-{[3-(2-methylphenyl)phenyl]methyl}pyrrolidine-2-carboxamide
7-(2,2-dimethylpropyl)-2-(5-ethyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3-fluorophenoxy)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidine
4-(3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-2-methylbutan-2-ol
5-(furan-2-yl)-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
3-(5-acetyl-2-methoxyphenyl)-1-(oxan-4-yl)urea
(2R,6S)-4-(6-chloro-3-{[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)-2,6-dimethylmorpholine
N-[4-(propan-2-yl)phenyl]-3-{[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amino}propanamide
6-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-methyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
(2S)-N2-cyclohexyl-N2-(pyridin-2-ylmethyl)pyrrolidine-1,2-dicarboxamide
5-methyl-1-propyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
9-(2-hydroxypyridine-3-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-6-(propan-2-yl)pyrimidine
4-(3-benzyl-1H-pyrazol-5-yl)-1-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
[4-(2,3-dihydro-1H-indene-5-carbonyl)-1,4-oxazepan-6-yl]methanol
(3R,4R)-1-cyclohexyl-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-ethyl-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
2-methyl-2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)propanamide
1-cyclohexanecarbonyl-4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(2-{1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
3-(1,2-oxazolidin-2-yl)-1-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}propan-1-one
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
6-(4-{[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)pyridine-3-carbonitrile