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5-{5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyridin-2-amine
(2,1,3-benzoxadiazol-5-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
4-{2-methyl-1-[4-(pyridin-3-yloxy)piperidin-1-yl]propan-2-yl}morpholine
1-{4-[2-(morpholin-2-yl)acetyl]piperazin-1-yl}-2-phenoxyethan-1-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}piperidin-2-one
(1S,5R)-3-(5-chlorothiophene-2-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-(1H-imidazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
3-[2-(2-methoxyethoxy)phenyl]-1-[1-(pyridin-3-yl)propan-2-yl]urea
1-{3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[9-(1H-imidazol-4-ylmethyl)-3-(1,3-thiazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-4-carbonitrile
methyl 4-(3-acetamidophenyl)-1H-pyrrole-2-carboxylate
2-[4-fluoro-3-(trifluoromethyl)phenyl]-N,N-dimethylbenzamide
6-[(4aR,8aR)-7-(dimethylcarbamoyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-5-chloropyridine-3-carboxylic acid
4-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-(4-methoxyphenyl)piperazin-2-one
(2S)-2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-4-methylpentan-1-ol
4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-methoxypyridine-3-carbonitrile
3-methyl-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
2-benzyl-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
[2-(azepan-1-yl)ethyl]({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(propan-2-yl)amine
1-[(4aR,8aR)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-6-yl]-2-methylpropan-1-one
5-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-1,3-benzothiazole
2-[1-ethyl-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]pyridine
2-ethyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N3,N3-diethyl-N1-(1H-indazol-5-yl)piperidine-1,3-dicarboxamide
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1,3,7-trimethyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-indole-2-carboxamide
3-{[ethyl(oxan-4-ylmethyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
1-ethyl-N-methyl-3-(2-methylpropyl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazole-5-carboxamide
N4-methyl-N2-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidine-2,4-diamine
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-9H-purin-2-amine
(4aS,8aS)-2-cyclohexyl-7-(2-methylpyrimidine-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-({4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}methyl)-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]propanamide
6-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
9-[(2S)-1-methylpyrrolidine-2-carbonyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-acetyl-5-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)methanesulfonamide
N-methyl-2-(methylsulfanyl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-7-methoxy-1-methyl-1,2-dihydroquinolin-2-one
3-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridazine