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2-(2H-1,3-benzodioxol-5-yl)-5-(pyrrolidin-1-ylmethyl)pyridine
3-{2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
5-[6-amino-5-cyano-4-(5-methylfuran-2-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)benzamide
N-tert-butyl-2-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]benzene-1-sulfonamide
methyl (2S,4R)-4-(3-chlorobenzamido)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidine-2-carboxylate
6-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-(hydroxymethyl)azepan-4-ol
1-[(5-ethylpyridin-2-yl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
{[(3S,4R)-1-(5-chlorothiophene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(4aR,8aR)-7-(5-ethyl-2-methylpyrimidin-4-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-{2-[4-(propan-2-yl)phenyl]ethyl}-1λ6-thiolane-1,1-dione
4-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-3-yl]benzoic acid
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
[3-(cyclopropylmethyl)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-yl]methanol
2-(4-methoxy-2-methylphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4,4-difluoropiperidine
N-[(1R,3R)-3-aminocyclopentyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1S,2S)-2-hydroxycyclohexyl]-3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzene-1-sulfonamide
5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-1-(4-methylphenyl)-1H-1,2,4-triazole
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4-methoxybenzamide
1-(1-benzoxepine-4-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
3-benzyl-3-[3-(1,4-diazepan-1-yl)-3-oxopropyl]-1-methyl-2,3-dihydro-1H-indol-2-one
N-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]morpholine-4-carboxamide
4-[7-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-(2-{[2-(2-chlorophenyl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
6-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]hexan-1-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-({5-[(3-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N3-benzyl-N5-ethyl-N3-methyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}phenol
(1R,5R)-3-(dimethylsulfamoyl)-N-(4-fluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(2-hydroxybutyl)-1H-pyrazole-4-carboxamide
N-(1-hydroxybutan-2-yl)-3-methyl-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
2-methoxy-5-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenol
N-[2-(dimethylamino)ethyl]-5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(4-phenylpiperidin-1-yl)methyl]-4-(pyridin-3-yl)phenol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[6-(piperidin-4-yl)pyrimidin-4-yl]piperazin-2-one
3-{2-[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
(3S)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methylpyridin-2-amine
8-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)azetidine-1-carboxamide
5-ethyl-1'-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-benzyl-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine