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3-{5-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
benzyl 3-{[(pyridin-2-ylmethyl)carbamoyl]methyl}morpholine-4-carboxylate
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
(2S,4S)-4-amino-N-{[2-(benzyloxy)phenyl]methyl}-1-methylpyrrolidine-2-carboxamide
4-phenyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenol
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-(1H-imidazol-1-yl)-1-(2-methyl-1-benzofuran-7-carbonyl)piperidine-4-carboxylic acid
5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
1-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(2-methyl-1,3-benzothiazol-6-yl)urea
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)pyridine-3-carboxamide
1-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}phenyl)-1H-1,2,4-triazole
N-(2-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]piperidin-3-yl}ethyl)acetamide
(2S,4S)-4-cyclohexaneamido-N-ethyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidine-2-carboxamide
(3S,4R)-1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
4-butyl-N-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]piperazine-1-carboxamide
3-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-2-yl}pyridine
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]prop-2-enamide
methyl (2S,4R)-4-[2-(1H-pyrazol-1-yl)benzamido]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
3-[2-(dimethylamino)ethyl]-8-(2-ethoxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,5R)-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2H-1,3-benzodioxol-5-yl)-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
3-({2-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(2R)-N-(adamantan-1-ylmethyl)-N-(2-hydroxyethyl)oxolane-2-carboxamide
1-(4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-(propan-2-yl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridine
1-(2-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(2S,4S,5R)-5-(2-chlorophenyl)-4-{[2-(dimethylamino)ethyl]carbamoyl}-1,2-dimethylpyrrolidine-2-carboxylic acid
3-[1-(3-chloro-2-fluorobenzoyl)piperidin-4-yl]-N-phenylpropanamide
6-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2,4-dimethylpyridine-3-carbonitrile
N-methyl-2-(oxan-2-ylmethoxy)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
5-(2-methylpropyl)-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(4-fluorophenyl)-2,2-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}cyclopropane-1-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-[(3-methoxyphenyl)amino]butanamide
4-ethyl-1-methyl-3-{[1-(quinolin-4-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
2-cyclopropyl-N-[(1-methylpiperidin-4-yl)methyl]acetamide
1-(2-{2-[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)piperidin-4-ol
7-chloro-2-methyl-4-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}quinoline
2-cyclohexyl-6-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-benzoxazole
4-{3-[(1-methanesulfonylpiperidin-4-yl)amino]butyl}phenol
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyridine-4-carboxamide
7-(1-benzyl-1H-pyrazole-4-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(1S,5R)-6-[3-(benzyloxy)propyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
4-(hydroxymethyl)-1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]azepan-4-ol
(2S,4S)-4-amino-1-methyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}pyrrolidine-2-carboxamide
(3R,4R)-4-cyclobutyl-N-(furan-2-ylmethyl)-4-hydroxy-3-methylpiperidine-1-carboxamide
2-amino-4-{[2-methoxy-2-(thiophen-2-yl)ethyl]amino}quinazoline-6-carboxylic acid