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N,N-dimethyl-4-oxo-4-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butanamide
1-(4-methylphenyl)-4-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]piperazin-2-one
N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
(3R,4R)-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(cyclohexylmethyl)-N,N-dimethyl-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-5,6-dimethylpyridine-3-carboxamide
ethyl[(2-methyl-2H-indazol-3-yl)methyl]{[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazo[1,2-b]pyridazine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[3-(furan-2-yl)propanoyl]piperidin-3-yl}propanamide
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
2-(furan-2-yl)-5-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]pyrimidine
(4aS,8aS)-2-[1-(methoxymethyl)cyclobutanecarbonyl]-7-(pyridin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-(3-chloro-4-fluorobenzoyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
8-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-4-[(dimethylamino)methyl]-N-(2-fluoro-4-methylphenyl)-3-hydroxypiperidine-1-carboxamide
5-(1H-imidazol-2-ylmethyl)-8-methoxy-2-[2-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-(pyrrolidin-1-yl)-3-[(trimethylpyrimidin-4-yl)amino]propan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2,2-dimethylpropyl)acetamide
1-(but-2-ynoyl)-N-[3-(3-chlorophenyl)phenyl]piperidine-4-carboxamide
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5,6,7,8-tetrahydroquinoline
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(3S,4R)-1-(1-benzofuran-2-ylmethyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-indazole
3-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-4,5,6,7-tetrahydro-2H-indazole
N3-ethyl-N3-{[3-(prop-2-en-1-yloxy)phenyl]methyl}piperidine-1,3-dicarboxamide
1-[4-(4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)phenyl]ethan-1-one
(1-{[methyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amino]methyl}cyclopropyl)methanol
4-(3-phenylpropyl)morpholine-2-carboxamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-5-methyl-1-benzofuran-2-carboxamide
3-methoxy-1-(2-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
2-(4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)-1,3-benzothiazole
(3S,4R)-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-methylpiperidine-3,4-diol
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-acetyl-N-(1-cycloheptylpiperidin-3-yl)piperidine-4-carboxamide
2-{[5-(3-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-methylacetamide
[(3-chloro-4-fluorophenyl)methyl](methyl)(oxan-2-ylmethyl)amine
N-cyclohexyl-N-(pyridin-2-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2,4-dimethyl-6-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyrimidine
(4aR,7aS)-1-(2-hydroxyethyl)-4-(4-methylpentyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(2,5-dimethylphenyl)methyl]urea
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(pyrimidin-2-yl)piperidin-4-ol
6-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
4-[5-(1-methyl-1H-pyrazol-4-yl)furan-2-carbonyl]morpholine
N-(adamantan-1-ylmethyl)-N-methyl-3-(2-oxooxolan-3-yl)propanamide
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
methyl (2R)-2-{[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}propanoate
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
2-[(2,3-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid