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2-[(1,3-benzothiazol-2-yl)amino]-N-[1-(3-methylpyridin-2-yl)ethyl]acetamide
6-[(diethylamino)methyl]-N-(6-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4-methyl-1,2,3-thiadiazole-5-carboxamide
2-methoxy-5-(1-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyrimidine
1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(quinazolin-4-yloxy)ethan-1-one
6,8-dimethyl-2-[({3-[(pyridin-3-yl)amino]propyl}amino)methyl]quinolin-4-ol
[5-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)furan-2-yl]methanol
1-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
1-[(3S)-3-ethylmorpholin-4-yl]-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
1-[2-({3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenyl]-4-methylpiperazine
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(2S,4S)-1-benzoyl-N-ethyl-4-(3,3,3-trifluoropropanamido)pyrrolidine-2-carboxamide
2-(4-fluorophenyl)-N-(oxan-4-yl)imidazo[1,2-a]pyridine-6-carboxamide
N-[(3R,4R)-1-[(5-acetylthiophen-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
3-{[(5-methylthiophen-2-yl)methyl]({[4-(pyrimidin-2-yloxy)phenyl]methyl})amino}propan-1-ol
2-methyl-4-{4-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}but-3-yn-2-ol
6-(5-methylfuran-2-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
3-methyl-6-(3,4,5-trimethoxyphenyl)pyridazine
[(3S,5R)-5-[(dimethylamino)methyl]-1-(1-phenylcyclopentanecarbonyl)piperidin-3-yl]methanol
5-methanesulfonyl-2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidin-4-amine
(2S,4R)-4-amino-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
2-{3-[1-methyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}pyridine
6-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-(methoxymethyl)-1-{[(1R,2R)-2-phenylcyclopropyl]methyl}pyrrolidine
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
2-(cyclopropylmethyl)-8-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-(3,4-dimethylphenyl)piperidin-3-amine
4-[3-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyridine
({5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-6-ylmethyl)benzamide
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
5-({[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
(1S,5R)-6-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-(2-oxopropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopentyl-N'-[2-(pyridin-4-ylformamido)ethyl]butanediamide
N-{[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
8-(1-ethyl-1H-pyrazole-3-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(propan-2-yl)-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
2-(4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)pyrimidine
3-[(3R,4S)-1-(4-methoxy-3-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
1-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-3-[(dimethylamino)methyl]piperidin-3-ol
(3S,9aR)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-(oxan-4-ylmethyl)piperidin-4-amine
4-({2-[1-(4-ethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[1-(4-tert-butylbenzoyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one