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ethyl 5-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-3-methylpyrazine
[2-(2,3-dihydro-1H-indol-1-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-(1-methyl-1H-pyrrol-2-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}-2-oxo-N-propylacetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[3-(methylcarbamoyl)pyrrolidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
1-methyl-4-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
2-[(4aR,7aS)-4-[3-(dimethylamino)benzoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
5-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}pyridin-2-amine
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
3-(2-hydroxyphenyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methylpyridine
8-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
9-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-phenylbenzoyl)-1-(thiophene-3-carbonyl)piperidine
2-benzyl-9-[2-(propan-2-ylsulfanyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-chlorophenyl)methyl]-2-oxo-6-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)-N-(5-oxo-1-propylpyrrolidin-3-yl)acetamide
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-chloro-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
2-({3-[(4-fluorophenyl)amino]piperidin-1-yl}methyl)phenol
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1,8-naphthyridine-2-carboxamide
ethyl 1-(7-chloroquinolin-4-yl)-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate
4-[3-cyclopropyl-5-(2-phenoxyethyl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
(1S,5R)-3-[5-(methoxymethyl)furan-2-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-fluoro-4-methoxyphenyl)-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}acetic acid
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
dimethyl({2-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-2-yl]ethyl})amine
N-(2-fluorophenyl)-3-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
2-(2-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
(1S,6R)-9-[3-(thiophen-3-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
methyl 2-{2-[(adamantan-1-yl)carbamoyl]acetamido}-4-(methylsulfanyl)butanoate
1-cyclohexanecarbonyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-{4-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-methylpyrimidin-2-yl}phenol
1-cyclohexyl-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-4-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-(propan-2-yl)-1-{2-[1-(pyridine-2-carbonyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-(5-acetamido-2-methoxyphenyl)-2-(hydroxymethyl)piperidine-1-carboxamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[3-(methylsulfanyl)phenyl]methyl}urea
2-[3-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,2,3-benzotriazole
(1R,5S)-6-methyl-N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N4-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane