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4-(hydroxymethyl)-N-[4-(2-methoxyphenoxy)phenyl]piperidine-1-carboxamide
4-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
N-ethyl-1-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
(2S,4R)-1-benzyl-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-N-methylpyrrolidine-2-carboxamide
2-oxo-N-(2-phenylethyl)-6-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
2-{[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
6-[(3-methoxy-2-propoxyphenyl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-2-(methoxymethyl)-6-methyl-1-(3-phenylpropyl)-1,4-dihydropyridin-4-one
2-({6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
2-[3-(3-cyanopiperidine-1-carbonyl)benzenesulfonamido]-N,N-dimethylacetamide
3-methyl-1-[1-(6-{[2-(pyridin-4-yl)ethyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
N-(pyrazin-2-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N'-(4-methylphenyl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)ethanediamide
2-(cyclopropylmethyl)-N-(3-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{4-[(1H-imidazol-2-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrrole-2-carboxamide
4-ethyl-6-{4-[3-(2-methoxyphenoxy)azetidin-1-yl]piperidin-1-yl}-2-methylpyrimidine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-methyl-1,3-oxazole-4-carboxamide
4-ethyl-3-(piperidin-4-ylmethyl)-1-(pyridin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
5-tert-butyl-4-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}furan-2-carboxamide
4-(3-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-3-oxopropyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-tert-butyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
3-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]aniline
methyl 2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-2-yl)acetamide
2-methyl-N-[2-(morpholin-4-yl)propyl]-6-(piperidin-4-yl)pyrimidin-4-amine
N-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-oxopropyl}methanesulfonamide
6-(3-chloro-5-fluorophenyl)-N,N-dimethylpyrimidin-4-amine
5-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-4-phenyl-1H-pyrazole-3-carboxamide
5-{4-[2-(adamantan-1-yl)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-methyl-N-(quinolin-6-ylmethyl)furan-3-carboxamide
1-[(3-methylphenyl)methyl]-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(1H-imidazol-2-yl)benzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
1-{4-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
3-({4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}methyl)-5-methyl-1,2,4-oxadiazole
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)acetamide
ethyl 1-{1-[1-(3-methylbutyl)-7-oxoazepan-4-yl]piperidin-4-yl}piperidine-3-carboxylate
(1S,5R)-6-methyl-3-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(2,3,4-trimethoxybenzoyl)morpholin-3-yl]acetic acid
6-(4-fluoro-2-methoxyphenyl)-N4,N4-dimethylpyrimidine-2,4-diamine
(3aS,6aS)-2-(cyclopropylmethyl)-5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
3-({[(3-hydroxyphenyl)methyl](methyl)amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one