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(3aS,6aS)-5-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
{7-[4-(4-methylpiperazin-1-yl)quinazolin-6-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-(quinolin-5-yl)piperidine-1-carboxamide
N-(furan-2-ylmethyl)-N-(2-methylpropyl)-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(1H-imidazol-2-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
4-{3-cyclopropyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-5-phenyl-1H-pyrazole
3,3-dimethyl-1-({5-[(3-methyl-1-benzofuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-(3,4-difluorophenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-amine
2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
1-(cyclopropylmethyl)-5-[2-(1H-indazol-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-(2,5-dimethoxyphenyl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
N-[(3R,4S)-1-(2-methanesulfonamidoacetyl)-4-phenylpyrrolidin-3-yl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-1-(propan-2-yl)piperidine-4-carboxamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-3-(4-hydroxyphenyl)-N-methylbenzamide
2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-propoxypiperidine
(3R,4R)-4-cyclobutyl-1-[(4-methoxypiperidin-1-yl)sulfonyl]-3-methylpiperidin-4-ol
2-(3-methoxypropyl)-8-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-4-yl)ethyl]amine
(1S,5R)-6-(cyclopropylmethyl)-3-(3-hydroxy-4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[4-({ethyl[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)phenyl]ethan-1-one
3-(3-hydroxybutyl)-5-methyl-3,4-dihydroquinazolin-4-one
1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidine-3-carbonitrile
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]butan-1-one
1-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-2-phenylethane-1,2-dione
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(4-phenylpiperidin-1-yl)acetamide
2-[4-(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)piperazin-1-yl]ethan-1-ol
ethyl 4-[(2-chlorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxylate
({5-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]pyridine-2-carbonitrile
2-(2-methylpropyl)-8-(2-oxoimidazolidine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
6-methyl-2-oxo-5-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridine-3-carbonitrile
2-{[3-(1H-imidazol-2-yl)-6-methoxyquinolin-2-yl]sulfanyl}acetic acid
N,1,3-trimethyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
8-benzoyl-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-fluorophenoxy)-1-(2-methylpyrimidine-5-carbonyl)piperidine-4-carboxylic acid
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
4-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-6,8-dimethyl-2H-chromen-2-one
4-[(2S)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidine-2-carbonyl]morpholine
N-[(3S,4R)-1-[2-(methylamino)pyridine-4-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-methyl-4-(3-{4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]piperidin-1-yl}phenyl)pyrimidine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4-hydroxyphenyl)-N-methylbenzamide
(2R,3S,6R)-5-(4-methyl-1H-imidazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-{8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carbonitrile
4-{1-[2-(pyridin-3-yl)acetyl]pyrrolidin-3-yl}benzoic acid