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N-(4-cyanophenyl)-4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]butanamide
1-[2-(1H-imidazol-2-yl)benzoyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
5-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
2-chloro-4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-6-methoxyphenol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methylpiperidine-2-carboxamide
N2-(2,1,3-benzoxadiazol-5-ylmethyl)-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
methyl 5-({2-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetamido}methyl)furan-2-carboxylate
1-methyl-4-(2-methyl-6-propylpyrimidin-4-yl)piperazine-2-carboxylic acid
3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenol
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-phenyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
7-chloro-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,3,5-trimethyl-1-benzofuran-2-carboxamide
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-fluorophenyl)-1,4-diazepane
2-(3-methoxypropyl)-9-(pyridine-3-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-methoxy-2-methylpropan-1-one
N-cyclopropyl-2-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidine
2-(2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethoxy)acetamide
5-phenyl-N-(4-{4-[(pyridin-4-ylmethyl)amino]piperidin-1-yl}phenyl)pentanamide
(3S,4S)-N-(4-cyanonaphthalen-1-yl)-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methyl-1,3-benzoxazole-6-carbonyl)piperidin-3-ol
(3S)-1,3-dimethyl-4-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperazin-2-one
5-(2,2-dimethyloxan-4-yl)-1-(4-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
N-(2-fluorophenyl)-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
5-methyl-1-{2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-2-[(2R)-5-oxopyrrolidine-2-carbonyl]-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-{4-[(2-hydroxy-7-methylquinolin-3-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
3-(2-hydroxyphenyl)-N-[1-(methoxymethyl)cyclopentyl]-1H-pyrazole-5-carboxamide
9-(2-ethylpyridine-4-carbonyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-[(3S,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(2-{1-[2-(morpholin-4-yl)butanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-methoxy-5-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}phenol
1-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-3-(1-methylpiperidin-3-yl)propan-1-one
N-[1-(4-methanesulfonylphenyl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
2-(4-fluorophenyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}acetamide
5-{1-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyridin-2-amine
{3-[(2,4-difluorophenyl)methyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl}methanol
N-(propan-2-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
3-(5-cyclobutyl-1H-1,2,4-triazol-3-yl)pyridine
3-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-6-methyl-1,2-dihydroquinolin-2-one
1-(6-carbamoylpyrazin-2-yl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
3-methyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
6-[3-(pyridin-4-yl)azetidin-1-yl]-9H-purine
4-cyano-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
1,3,6-trimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
7-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroquinoxalin-2-one
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-(1,3-thiazol-2-ylmethyl)imidazolidine-2,4-dione
1-(2-aminoethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide