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1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-3-(3-methoxy-4-methylphenyl)propan-1-one
(3R,4S)-4-cyclopropyl-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-amine
1,3-dimethyl-N-[2-(6-methylpyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N,N-dimethyl-5-[4-(piperidin-1-yl)butanoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(3R,4R)-3-cyclobutyl-4-methyl-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
2-(1H-imidazol-2-yl)-N-[3-(1H-indol-1-yl)propyl]benzamide
(1S,5R)-3-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
3-{[1-(3-methanesulfonylbenzoyl)piperidin-4-yl]methyl}benzoic acid
4-({2-[1-(cyclopropanesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(1R,5R)-6-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4R)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-(3-{3-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
(4aR,8aR)-7-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-(3-hydroxyadamantan-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
5-(3-methoxyphenoxymethyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
6-(1,4-oxazepan-4-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
1-ethyl-3-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indazole
(3S,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
methyl 3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
1-(cyclobutylmethyl)-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxypiperidin-2-one
ethyl 4-[3-(1-acetamido-3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]piperidine-1-carboxylate
4-[4-(5-hydroxypyrazine-2-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
3-methyl-8-[2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-{[(1R)-1-phenylethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
({4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
1-[3-chloro-2-(propan-2-yloxy)phenyl]-3-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]urea
2-methyl-5-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]quinoline
4-[(1-{[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
8-benzyl-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}sulfonyl)benzoic acid
3-cyclopentyl-1-{2-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}propan-1-one
1-(carbamoylmethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
4-[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1-phenylbutan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrimidin-4-ol
(benzylsulfamoyl)({[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](1-phenoxypropan-2-yl)amine
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-hydroxypropyl)acetamide
1-methyl-4-({6-[(1E)-pent-1-en-1-yl]pyridin-3-yl}methyl)piperazine
2-methyl-7-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aR,8aS)-1-(cyclopent-1-ene-1-carbonyl)-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
6-(1-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
7-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-oxa-7-azaspiro[3.5]nonane
methyl (2R,4S)-1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-hydroxypiperidine-2-carboxylate
N,1-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine