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N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-(morpholine-4-carbonyl)piperidine-1-carboxamide
[(3aS,6aS)-2-(6-ethyl-2-methylquinoline-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
3-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-cyclohexyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
1-[(2-chlorophenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(4aS,8aR)-6-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
2,6-dihydroxy-N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-4-(1H-pyrazol-4-yl)butanamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-methoxy-1-methyl-1H-indole-2-carboxamide
2-[5-(4,6-dimethylpyridin-3-yl)-1-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]acetamide
3-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}quinoline
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(3-methylthiophen-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
N-(2-hydroxy-2-phenylethyl)-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(piperidin-1-ylmethyl)piperidine
2-(5-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[3-(methylsulfanyl)propyl]amine
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
3-phenoxy-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(2S,4S,5R)-1-methyl-4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(oxolan-3-yl)piperidine-4-carboxamide
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-benzyl-N-(3,4-difluorophenyl)piperidin-3-amine
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(4-methoxybenzoyl)piperazine
5-acetyl-2,4-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrrole-3-carboxamide
5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
N-methyl-N-(thiophen-3-ylmethyl)-1-benzofuran-3-carboxamide
2-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-amine
1-(1,3-dihydro-2-benzofuran-5-yl)-3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)urea
(2S)-1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-methyl-2-(propan-2-yl)piperazine
7-[(2,3-dimethoxyphenyl)methyl]-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
8-(2-ethylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
2-methoxy-1-[1'-(2-methyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(3R,5S)-5-[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol
6-[3-(butylcarbamoyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1R,5R)-3-benzoyl-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(2-methyl-1,3-thiazol-4-yl)-1-[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
[(1-cyclopentylpiperidin-3-yl)methyl][(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl][2-(piperidin-1-yl)ethyl]amine
N-[3-(1,3-benzoxazol-2-yl)propyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-[(3-chlorophenyl)methyl]-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-3-carboxylic acid
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
8-[(4-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[1-(pyridin-4-yl)propyl]benzamide
(1S,5R)-3-[(3-methylquinoxalin-2-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
dimethyl(2-{[(6-methylpyridin-2-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)amine