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1-(furan-3-carbonyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
(2S,4S,5R)-5-(4-chlorophenyl)-4-[(2-hydroxyethyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
3-(4-hydroxyphenyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
(4aS,7aR)-1-[(2,6-dichlorophenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-methoxypropyl)-1-(3-methylthiophene-2-carbonyl)piperidine-3-carboxylic acid
2-(3-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-2-methyl-1H-indol-1-yl)acetic acid
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
5-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}methyl)-N-methylpyrimidin-2-amine
(3S)-1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-ol
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(pyrazin-2-yl)acetamide
2-[5-(2,4-difluorophenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-methoxyphenoxy)-2-methylpropan-1-one
1-cyclopropanecarbonyl-N-{[1-(2-fluorophenyl)cyclopentyl]methyl}piperidine-4-carboxamide
{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-[(1R,3R)-3-aminocyclopentyl]-4-(4-ethoxy-3-methylphenyl)-4-oxobutanamide
8-(5-phenylpentanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
6-(2,5-dimethylfuran-3-yl)-N,N-dimethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrrol-1-yl)pyridine
3-[(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
1-cyclohexyl-N3-(cyclohexylmethyl)-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperidin-4-yl}methanesulfonamide
2-[4-({[(1R,2S)-2-(methoxymethyl)cyclopentyl]carbamoyl}amino)phenyl]-N-methylacetamide
5-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)-N,N-dimethylpyridin-2-amine
N-[(1-{3-[4-(dimethylamino)phenyl]propanoyl}piperidin-4-yl)methyl]acetamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-(morpholine-4-sulfonyl)benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,4-dithiepan-6-amine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-chloro-1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-5-(cyclopropylmethyl)-8-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
ethyl 4-[2-(1-phenylethyl)-1H-imidazol-1-yl]piperidine-1-carboxylate
2-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]pyrimidin-4-amine
(3S,4S)-4-methyl-1-[2-(methylamino)pyridine-3-carbonyl]piperidine-3,4-diol
methyl 2-({4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)-4-(methylsulfanyl)butanoate
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}quinoxaline-5-carboxamide
2-acetyl-8-[2-(phenylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{2-[1-(1H-imidazol-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-1-phenylurea
(1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2,5-dihydro-1H-pyrrole
2-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
3-(5-methyl-1H-pyrazol-1-yl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
4,4-difluoro-1-{[5-(1,2,5-thiadiazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(3-methyl-2-oxoimidazolidin-1-yl)acetamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
6-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
N-methyl-4-(1H-pyrazol-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
N-[2-(benzyloxy)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-methyl-5-propyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine