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1-[4-(3-fluorophenyl)phenyl]-3-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methylurea
[4-benzyl-1-(3-ethyl-1H-indole-2-carbonyl)piperidin-4-yl]methanol
2-(6-methoxypyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-methyl-N-{2-phenyl-1-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl}thiophene-3-carboxamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-phenylacetamide
5-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile
1-[(4-chlorophenyl)methyl]-5-[4-(hydroxymethyl)piperidine-1-carbonyl]piperidin-2-one
4-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}benzoic acid
5-(2-aminopyrimidin-4-yl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[(5-chlorothiophen-2-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
(2S)-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
2-chloro-N-{1-[1-(2-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-(4-{[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]amino}piperidin-1-yl)butan-1-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
3-(benzyloxy)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
methyl 3-(2-methylbutanamido)-5-[(2-methylpropyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(5-ethylpyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
1-[(5-{[4-(2-hydroxyethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3,4-dimethoxyphenyl)-2-[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
3-(2,5-dimethoxyphenyl)-4-methylbenzamide
5-(1H-imidazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-methoxy-5-oxo-6-[(2R)-oxolan-2-ylmethyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
11-[(3,4-dimethylphenyl)methyl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenol
(3R,5R)-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
4-[(2-chloro-5-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[3-(4-ethylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,6-dimethyl-2H-pyran-2-one
1-{3-[3-(2-fluorophenoxy)azetidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(3-methoxypiperidin-1-yl)-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidine
[(3R,4R)-1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-hydroxy-2-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]benzamide
2-{4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrazine
3-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazol-5-yl}-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
(4aS,7aR)-1-(3-methoxy-2-methylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,7aS)-2-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-cyclopropanecarbonyl-1'-{imidazo[1,2-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
5-{1-[(5-fluoro-2-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}-8-methylquinoline
2-(ethanesulfonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
N-{4-chloro-3-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]phenyl}acetamide
2-phenyl-1-(1-{2-[(prop-2-en-1-yl)amino]benzoyl}piperidin-4-yl)ethan-1-ol
methyl 2-hydroxy-5-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}benzoate
1-(2,3-difluoro-6-methoxybenzoyl)-3-(2,6-dimethylphenoxy)azetidine
2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
5-(2,4-dimethylphenyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazole