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(1S,5R)-6-[(1-ethyl-1H-indol-4-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-(2,3-dimethylquinoxalin-6-yl)-1-[3-(morpholin-4-yl)propyl]urea
6-(4-methanesulfonylpiperazin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
5-[3-({[ethyl(methyl)sulfamoyl]amino}methyl)pyrrolidin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine
(3S,4S)-4-{[({3-[3-(trifluoromethyl)phenoxy]phenyl}methyl)amino]methyl}piperidin-3-ol
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-[4-(2-propyl-1H-imidazol-1-yl)phenoxy]ethan-1-ol
1-(morpholin-4-yl)-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
1-[2-(pyridin-4-yl)-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
(2S)-1-acetyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyrrolidine-2-carboxamide
2-[(E)-2-cyclohexylethenyl]-5-(pyrrolidine-1-carbonyl)pyridine
1-[(3-chloro-5-fluorophenyl)methyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[2-({1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}amino)pyrimidin-4-yl]piperidin-4-ol
2-{4-[(3-ethenylphenyl)methyl]piperazin-1-yl}-5-fluoropyrimidine
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxylate
1-{7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}-3-phenoxypropan-1-one
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
4-(cyclohexylmethyl)-3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(2-methylfuran-3-carbonyl)piperidine
4-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
(2R,3R,6R)-5-(2,5-dimethylbenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(diphenylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-methyl-6-oxo-N-[1-(pyridin-4-yl)propyl]-1,6-dihydropyrimidine-5-carboxamide
(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]pyrrolidin-3-amine
2-cyclopropyl-4-phenyl-9-propanoyl-2,9-diazaspiro[5.5]undecan-3-one
2-(azepan-1-yl)-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}acetamide
7-chloro-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidine-2-carboxamide
N-{4-[({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)methoxy]phenyl}furan-2-carboxamide
N1,N1,N4-trimethyl-N4-(quinolin-5-ylmethyl)piperidine-1,4-dicarboxamide
3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(4-fluorophenyl)methyl]-5-(2,4,5-trimethylbenzoyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(pyrrolidine-1-carbonyl)piperazine
1-{[5-({4-[1-(dimethylamino)ethyl]phenyl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
N-[(3S,4R)-1-(4-cyanopyridin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-(dimethyl-1,3-thiazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(1,2-benzoxazol-3-yl)-N-[(2-chloropyridin-3-yl)methyl]-N-methylacetamide
1-[(4-methylphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-{[2-(3,4-dimethylphenoxy)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-methyl-3-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
2-{2-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amine
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetic acid
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
3-methoxy-N-(4-sulfamoylphenyl)piperidine-1-carboxamide