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N-[(3S)-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl]acetamide
3-({methyl[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)phenol
1-[(3-chloro-2-fluorophenyl)methyl]-3-(1-methyl-1H-1,2,4-triazol-3-yl)urea
2-[5-(3-methoxyphenyl)furan-2-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[3-(oxolan-2-yl)propyl]pyrimidine-5-carboxamide
4-(1-benzofuran-2-yl)-N,N-dimethylbenzamide
6-chloro-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}imidazo[1,2-a]pyridine-2-carboxamide
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(oxolan-2-ylmethyl)acetamide
N-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}methanesulfonamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
1-[1-(3-methoxybenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
4-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-6-ethyl-1,2-dihydropyridin-2-one
3,5-dimethyl-4-(5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)-1,2-oxazole
4-({2-[1-(difluoromethyl)-3-methyl-1H-pyrazol-4-yl]phenyl}methyl)morpholine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-phenylethyl)piperidine-4-carboxamide
N-ethyl-N-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}oxan-4-amine
1-(4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
4-[hydroxy(thiophen-2-yl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
3-(4-{3,9-diazaspiro[5.6]dodecan-9-yl}-4-oxobutyl)-3,4-dihydroquinazolin-4-one
5-fluoro-2-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-{2-[(4-chloro-1-methyl-1H-pyrazol-3-yl)formamido]ethyl}pyridine-3-carboxamide
2-({ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzoic acid
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(methanesulfonylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazole
(4S,4aS,8aS)-1-(5-hydroxypyrazine-2-carbonyl)-4-phenyl-decahydroquinolin-4-ol
4-ethyl-3-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(azepan-1-yl)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}propan-2-ol
1-{2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
(1S,2S)-2-{4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)(quinolin-2-ylmethyl)amine
2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-1H-indole
5-[(3-methyl-3-phenylpiperidin-1-yl)methyl]pyrimidine
1-ethyl-4-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]-1H-pyrrole-2-carbonitrile
6-[(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]pyridine-2-carboxylic acid
1-(2-methylphenyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
3-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-N-(2,4-dimethylphenyl)-3-oxopropanamide
N4-ethyl-N2-[(5-methylpyrazin-2-yl)methyl]pyrimidine-2,4-diamine
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-1,3-thiazole-4-carboxamide
3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
7-fluoro-4-(6-methoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(pyrimidin-5-yl)quinoline
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
1-(4-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)ethan-1-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-(2-methoxyethyl)acetamide
(3S,4R)-1-(2-acetamido-2-methylpropanoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-{5-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
5-(3-chlorophenyl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1,2,4-triazin-3-amine
2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-ethyl-N-methylacetamide
1-(diethylamino)-3-[2-methoxy-4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propan-2-ol
1-{4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-1H-pyrazole
N-cyclopropyl-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-4-carboxamide