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1-[(2-methoxyphenyl)methyl]-4-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]pyrrolidin-2-one
1-(2-chlorobenzenesulfonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
3-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-(2-{[(4-hydroxy-6-methylquinolin-2-yl)methyl]amino}ethyl)acetamide
[1-(9H-fluoren-2-ylmethyl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
2-{3-[({[2-(1H-imidazol-1-yl)phenyl]methyl}amino)methyl]-2-methyl-1H-indol-1-yl}acetamide
3-{[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2,5-oxadiazole-3-carboxamide
2-{9-[(3-cyanophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-(furan-2-ylmethyl)-3-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-4-ylmethyl)propanamide
5-tert-butyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1,3,4-oxadiazol-2-amine
1-methyl-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(3-ethoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-(benzyloxy)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]butan-1-one
7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
(3S)-3-ethyl-4-[2-(4-fluorophenoxy)ethanesulfonyl]morpholine
1-cyclobutanecarbonyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
N-[2-(2-fluorophenyl)ethyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
N-(3,5-dimethylphenyl)-2-oxo-2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
4-(3,6-dimethylpyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(3-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}propyl)-1,2,5-oxadiazole-3-carboxylic acid
1-[(1S)-1-[3-(4-tert-butylphenoxymethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]ethyl]-1H-1,2,3,4-tetrazole
1-(4-carbamoyl-1,3-thiazol-2-yl)-4-phenoxypiperidine-4-carboxylic acid
2-[4-(methylsulfanyl)phenyl]-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{3,4-dihydrospiro[1-benzopyran-2,1'-cyclopentane]-4-yl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)piperidin-4-ol
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-[2-(diethylamino)ethyl]propanamide
2-(5-{imidazo[1,2-a]pyridin-2-yl}-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl)acetic acid
N-{2-[7-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
N5-butyl-1-cyclohexyl-N3-methyl-4-oxo-N3-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3aS,6aS)-2-benzyl-5-[2-(thiophen-2-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-amino-4-(4-hydroxynaphthalen-1-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2,2-dimethyl-5-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)pentan-1-ol
1-[(4-fluorophenyl)methyl]-4-(4-methyl-1,3-thiazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 6-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)pyridine-2-carboxylate
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1H-pyrrole-3-carboxamide
3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4-(pyridin-3-ylmethyl)piperazin-2-one
4-(2,2-diphenylethyl)-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
2-{4-[6-amino-5-cyano-4-(2-methoxyphenyl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]propanamide
(3S,4R)-4-phenyl-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidine-3-carboxylic acid
1-methyl-4-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carbonyl)piperazine
4-(4-fluorophenyl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1,2,3,6-tetrahydropyridine
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-[1-(thiophen-2-yl)propyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid