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3-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(benzenesulfonyl)piperidin-4-yl]-2-methyl-1,3-thiazole-4-carboxamide
5-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
4-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}azepane
{2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}urea
1-[(3-{[1-(furan-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
2-{4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
9-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-{[(1-ethylpyrrolidin-2-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
2-(2-phenylethyl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}morpholine
N-(1-cycloheptylpiperidin-3-yl)-3,5-dimethoxybenzamide
N-[(3-chlorophenyl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N,N-dimethyl-5-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridin-2-amine
1-[(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-(3-methoxypropyl)-N-(4-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
2-[(3-{[4-(oxolan-2-yl)butyl]carbamoyl}phenyl)amino]acetic acid
5-benzyl-3-[2-(pyridin-2-yl)ethyl]-5-[1-(thiolan-3-yl)piperidin-4-yl]imidazolidine-2,4-dione
7-[2-(4-methylbenzoyl)benzoyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
N-ethyl-2-[4-(3-hydroxyphenyl)piperazin-1-yl]pyridine-3-carboxamide
1-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-2-methyl-1,4-dihydroquinolin-4-one
1-(3-chloro-4-methoxyphenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-5-oxopyrrolidine-3-carboxamide
1-[2-(4-fluorophenyl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
N-{[2-(3-fluoro-4-methoxyphenyl)phenyl]methyl}propanamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[4-(furan-2-ylmethoxy)phenyl]urea
(1S,5R)-6-benzyl-3-[2-(dimethylamino)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2-chlorophenyl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(2-methylpropyl)acetamide
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
N,2-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[(pyridin-3-ylmethyl)amino]benzamide
N-[(3R,5S)-1-[(cyclopropylcarbamoyl)methyl]-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
1-[5-(2,5-dimethylphenyl)-1,2,4-oxadiazol-3-yl]-2-methylpropan-2-ol
1-{2-[5-(piperidine-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
5-(5-methylfuran-2-yl)-N-[3-(pyridin-3-yl)propyl]-1,2,4-triazin-3-amine
5-chloro-N-methyl-6-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,6-dihydropyridine-3-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-(4-{2-[methyl(piperidin-4-yl)amino]acetyl}piperazin-1-yl)-2-phenoxyethan-1-one
2-[2-({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]-1,2-dihydrophthalazin-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-hydroxyethan-1-one
5-methyl-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-cyclopentyl-2-methyl-N-(thiophen-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
(3S,9aR)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{2-[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione