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4-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)-1,3-thiazol-2-amine
2,2-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl}propan-1-one
2-[methyl(2-phenylethyl)amino]-N-(piperidin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(methylsulfanyl)ethyl]amine
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[2-(pyridin-4-yl)ethyl]benzamide
4-(3-ethoxy-4-methoxyphenyl)-5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-methyl-1-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinazolin-2-one
2-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
3-(5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
2-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl(2-phenylethyl){[3-({1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-(furan-2-yl)azepane
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2-methoxypyridine
({5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-methoxyphenyl}methyl)(methyl)amine
6-cyclopentyl-2-methoxy-3-({[5-(propan-2-yl)pyrimidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(3,4-dimethylphenyl)-1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-amine
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-[4-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]morpholine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
1-(6-chloro-3-{[3-(methoxymethyl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)azocane
N-[(5-ethylpyridin-2-yl)methyl]-1H-indazol-5-amine
4-{[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzamide
(4aR,8aR)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidin-2-one
3-(2-methoxyethyl)-1-[2-(thiophen-2-yl)acetyl]piperidine-3-carboxylic acid
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrimidin-2-amine
ethyl 1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-9-oxa-2-azaspiro[5.5]undecane
2-{4-[(3,4-dimethoxypyridin-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[1-(6-methylpyridin-2-yl)propan-2-yl]piperidine-4-carboxamide
ethyl 2-[4-(5-propylpyrimidin-2-yl)piperazin-1-yl]acetate
(2S)-4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}-2-hydroxybutanoic acid
3-cyclohexyl-5-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,2,4-oxadiazole
(1S,5R)-3-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N,4-trimethyl-3-({[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(benzylsulfamoyl)[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amine
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})methylamine
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
(1S,6R)-N-[2-ethoxy-5-(trifluoromethyl)phenyl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
2-(2-chlorophenyl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
2-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
N4-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
3,3-diphenyl-1-[(2R)-pyrrolidine-2-carbonyl]piperidine
3-[(1-{[4-(2-hydroxyethoxy)phenyl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
(2S,4S)-4-amino-1-[2-(2-chlorophenoxy)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
5-(morpholin-4-ylmethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide