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2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(piperazin-1-yl)acetamide
2-(dimethylamino)-N-[2-methyl-3-({[2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)phenyl]acetamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-methoxypyridine-3-carbonitrile
1-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-4-(cyclopropylmethyl)-1,4-diazepan-5-one
N-({4-hydroxy-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]azepan-4-yl}methyl)methanesulfonamide
1-(5-methoxy-2-methylphenyl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
N-cyclopropyl-5-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
8-methoxy-2-methyl-5-[1-methyl-5-(morpholin-4-yl)-1H-1,2,4-triazol-3-yl]quinoline
4-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[4-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
8-fluoro-2-({[(3S)-piperidin-3-yl]amino}methyl)quinolin-4-ol
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)(quinolin-5-ylmethyl)amine
5-[({[3-(2-methoxyethoxy)phenyl]carbamoyl}amino)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-{1-[(4-methanesulfonylphenyl)methyl]azetidin-3-yl}pyridine
2-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[3-(4H-1,2,4-triazol-4-yl)propyl]propanamide
3-[2-(4-fluorophenyl)ethyl]-1-(3-fluoropropyl)piperidine
N-[5-(2,4-dimethoxyphenyl)quinolin-8-yl]acetamide
2-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrazine
{2-[4-(5-chlorothiophene-2-carbonyl)morpholin-2-yl]ethyl}dimethylamine
[2-(2-ethoxyphenoxy)ethyl][(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
6-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
5-butyl-1'-(4-methyl-1,3-thiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cyclopentyl-4-{[(3-methoxypyrazin-2-yl)amino]methyl}pyrrolidin-2-one
4-ethyl-3-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-3-yl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-fluoro-3-methylphenyl)-2-[methyl(prop-2-yn-1-yl)amino]acetic acid
N-(trimethyl-1H-pyrazol-4-yl)-2,3-dihydro-1H-isoindole-2-carboxamide
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylpropanamide
4-[(dimethylamino)methyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)azepan-4-ol
N-[2-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3-(1-ethyl-5-oxopyrrolidin-3-yl)-1-[4-(4-methylphenyl)phenyl]urea
4-[(2E)-3-phenylprop-2-en-1-yl]-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{1-[1-(methoxymethyl)cyclopentyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-{[5-(2-fluorophenyl)furan-2-yl]methyl}-octahydropyrrolo[1,2-a]piperazine
(3R,9aR)-8-(4-chlorobenzoyl)-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
2-methyl-8-[3-(thiophen-3-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-{2-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-(1-propanoylazepan-3-yl)-4-(1H-pyrazol-1-yl)benzene-1-sulfonamide
2-[2-({cyclohexyl[2-(ethylsulfanyl)ethyl]amino}methyl)phenoxy]acetic acid
N-(1-hydroxybutan-2-yl)-N'-methyl-N'-phenyl-N-(pyridin-2-ylmethyl)ethanediamide
methyl 3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate