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N-{4-[(2-methyl-1,4-oxazepan-4-yl)methyl]phenyl}acetamide
3-ethoxy-4-(prop-2-en-1-yloxy)-N-[1-(pyridin-4-yl)propan-2-yl]benzamide
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-[(5-methylfuran-2-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
[(3,4-dimethoxyphenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-{3-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-4-methylbenzamide
methyl 4-(5-methyl-4-{[methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]methyl}-1,3-oxazol-2-yl)benzoate
(1S,5R)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-1-[4-(2-methanesulfonylethyl)piperazin-1-yl]-2-(4-methylphenyl)ethan-1-one
2-(3-fluoro-4-hydroxyphenyl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-(4-cyclopentyl-1,4-diazepan-1-yl)ethan-1-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(methylsulfanyl)phenyl]methyl})amine
4-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]sulfonyl}-2,1,3-benzothiadiazole
1-{[2-(2-methoxypyridin-3-yl)phenyl]methyl}piperazine
2-methyl-5-{4-[2-(pyrrolidin-1-yl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-({5-chloro-2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidine-3-carbonitrile
N-(2-chlorophenyl)-3-[1-(6-oxopiperazine-2-carbonyl)piperidin-4-yl]propanamide
1-({3-[3-(dimethylamino)propoxy]phenyl}methyl)azetidin-3-ol
5-({[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]carbamoyl}amino)-2-methoxybenzamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
6-(oxan-4-yl)-3-[(E)-2-phenylethenyl]-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-phenylpiperidine-4-carbonitrile
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-(1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1H-1,2,3-benzotriazole-5-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3-(methylsulfanyl)propanamide
1-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}-N-(3-methyl-1,2-thiazol-5-yl)benzamide
4-cyclopentyl-N-methyl-N-[2-(morpholin-4-yl)propyl]pyrimidin-2-amine
8-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,3-dimethoxy-5-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-(5-methyl-4H-1,2,4-triazol-3-yl)-N-(oxolan-3-ylmethyl)aniline
4-(3-fluorophenoxy)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidine-4-carboxylic acid
(3aR,5R,6S,7aS)-2-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
8-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-5-phenylpentan-1-one
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
1-cyclopropanecarbonyl-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]piperidine
4-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
4-[2-(2,3,6-trifluorophenyl)ethyl]-1λ6-thiomorpholine-1,1-dione
N-[4-(4-chlorophenoxy)phenyl]-3-(dimethylamino)pyrrolidine-1-carboxamide
3-[(2-methoxyethyl)sulfamoyl]-5-(quinolin-3-yl)benzoic acid
N-[2-(ethanesulfonyl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2,2-diethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-[N-benzyl-1-(8-fluoroquinolin-2-yl)formamido]propanamide
3-cyclohexyl-4-{[4-(1-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
3-[3-({[(4-phenyloxan-4-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
1-(1-benzothiophen-3-ylmethyl)-3-methylpiperidine-3-carboxamide