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1-(2-methyl-1-benzofuran-5-carbonyl)piperidine-2-carboxylic acid
N-benzyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-{1-[(5-chloro-2,4-dimethoxyphenyl)methyl]piperidin-2-yl}acetic acid
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-(2-methoxyphenyl)acetamide
4-ethyl-3-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]furan-2-carboxamide
(3R,4S)-4-cyclopropyl-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-amine
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
[4-({[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}methyl)oxan-4-yl]methanol
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-(4-chloro-3-methylphenoxy)-3-[(1-cyclopropylpropan-2-yl)amino]propan-2-ol
5-{4-[(1E)-pent-1-en-1-yl]phenyl}-1H-1,2,3,4-tetrazole
N-methyl-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-[2-(methylsulfanyl)ethyl]acetamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2,3,5,6-tetramethylbenzamide
7-(2-methoxyethyl)-2-[3-(2-methylphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
4-ethyl-3-{1-[(3E)-4-phenylbut-3-enoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,6R)-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-(2-methoxyethyl)-N-[3-(2-phenylacetamido)phenyl]pyrrolidine-3-carboxamide
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
N-(3-methoxyphenyl)-3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}propanamide
3-[(3R,4S)-4-(dimethylamino)-1-[4-(2-methylpropyl)benzoyl]piperidin-3-yl]propanoic acid
N-methyl-4-(1H-pyrazol-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)butanamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(quinoxalin-2-ylmethyl)pyridin-2-amine
2-(3-hydroxypropyl)-8-(1-phenylcyclopropanecarbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,6-dimethylpyrimidine-4-carboxamide
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(2-hydroxyethoxy)ethyl]acetamide
1-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carbonyl}-4-(hydroxymethyl)piperidin-4-ol
4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-2-(propan-2-yl)pyrimidine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(3,4-difluorophenyl)-5-{1-[(2,6-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-1-benzofuran-2-carboxamide
methyl[1-(1,2-oxazol-3-yl)ethyl]{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]quinoxalin-2-amine
N-[2-(oxan-2-yl)ethyl]-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-{2-[(6-phenylpyridazin-3-yl)oxy]hex-5-en-1-yl}morpholine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-phenylethyl)piperidin-3-ol
1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
1-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-(2-methylbutyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-(1-benzothiophen-2-ylmethyl)-11-{[(5-methylpyrazin-2-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-2-[methyl(piperidin-4-yl)amino]acetamide
3-benzyl-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
(1S,6R)-N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
2-(3-hydroxyphenyl)-2-[4-(2-methoxyethoxy)piperidin-1-yl]acetic acid