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N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1-methyl-1H-pyrazol-4-amine
N-[(4-methoxyphenyl)methyl]-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(3-fluorophenyl)-5-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
14-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(1S,2R)-2-({[6-(dimethylamino)pyridin-3-yl]methyl}(methyl)amino)cyclohexan-1-ol
2-{3-cyclopentyl-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-[3-(2,3-dihydro-1H-indol-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(2,1,3-benzoxadiazol-4-ylmethyl)({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)butanamide
1-methyl-4-[(2-{[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]oxy}phenyl)methyl]piperazine
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[(2-methyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]cyclobutanecarboxamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1-methylazepane-2-carboxamide
5-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R,6S)-2,6-dimethyl-4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
2-[1-(quinolin-2-ylmethyl)pyrrolidin-2-yl]ethan-1-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-ylmethyl)benzamide
N-benzyl-3-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-N-methylpropanamide
2-(1H-imidazol-2-yl)-1-(3,4,5-trimethoxyphenyl)-1H-imidazole
N-cyclopropyl-1-{2-[1-(3,3-dimethylbutanoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[(3R,4S)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-(4-phenylbutyl)acetamide
N-(1H-1,2,3-benzotriazol-4-yl)-2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-[2-(morpholin-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N,1-diethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}piperidine-2-carboxamide
5-(2,3-dimethylquinoxaline-6-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
methyl 3-benzamido-5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[4-(ethylamino)pyrimidin-2-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
5-(2-chlorophenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}furan-2-carboxamide
2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}thieno[3,2-d]pyrimidin-4-amine
11-[1-(azepan-1-yl)-2-methylpropan-2-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
4-{4-[4-(methylamino)pyrimidin-2-yl]piperazin-1-yl}butan-1-ol
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
4-chloro-N-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
2-(pyrrolidin-1-yl)-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-amine
3-cyclopropyl-5-{imidazo[1,2-a]pyridin-6-yl}-1-phenyl-1H-1,2,4-triazole
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
2-[1-(2-methylpropyl)-4-{[4-(propan-2-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
{[(1R,5S,6S)-3-(1H-1,3-benzodiazole-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[2-(methylsulfanyl)phenyl]urea
2-[4-(propan-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
4-hydroxy-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-phenylpyrimidine-5-carboxamide
N-[1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]-1-(pyridin-3-ylmethyl)piperidin-4-amine
N-(2-methoxyethyl)-1-methyl-N-(thiophen-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide