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N-[2-(benzyloxy)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]propanamide
N-(2-chloro-6-methylphenyl)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
5-[2-(3-methyl-1,2,4-oxadiazol-5-yl)phenoxy]-1-azabicyclo[3.2.1]octane
N-butyl-3-{[(3,5-dimethoxyphenyl)formamido]methyl}piperidine-1-carboxamide
ethyl 4-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperazine-1-carboxylate
(4aS,7aR)-1-(4-methylpyridine-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(4-acetylphenyl)methyl]-2-(pyridin-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-({5-[(2-butyl-1H-imidazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
N-{[7-(2-methoxy-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
8-butyl-N-(4-fluorophenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one
N-[(2,3-dimethoxyphenyl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
(4aS,8aR)-2-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-decahydroisoquinoline
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidin-4-amine
(3S,4S)-4-(4-fluorophenyl)-1-[(2-methoxypyridin-3-yl)methyl]piperidin-3-ol
(but-2-yn-1-yl)({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(furan-2-ylmethyl)amine
(2S)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-oxopyrrolidine-2-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
2-(dimethylamino)-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
1-(2,5-dihydro-1H-pyrrol-1-yl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
{1-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)methyl]cyclopropyl}methanol
N-(1-methoxypropan-2-yl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(6-methoxynaphthalene-2-carbonyl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-{3-[4-(4-formyl-1,4-diazepan-1-yl)piperidin-1-yl]phenyl}-2-methoxybenzamide
[(5-chloro-2-methoxyphenyl)methyl](ethyl){[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
(3R,5S)-N-(naphthalen-2-ylmethyl)-1-(pyridin-4-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
5-methyl-1-propyl-N-{[3-(trifluoromethoxy)phenyl]methyl}-1H-pyrazole-4-carboxamide
2-amino-8-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
6-({5H,6H,7H-cyclopenta[b]pyridin-7-yl}amino)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(piperidin-3-yl)benzamide
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-(4-methoxy-2-methylphenyl)propanamide
7-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(2S,4S)-4-amino-1-[1-(2-chlorophenyl)piperidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
5-acetyl-N,2,4-trimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrrole-3-carboxamide
3-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-1H-pyrazol-5-amine
4-(cyclopentylamino)-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
3-(1H-indol-3-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
6-oxo-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]piperazine-2-carboxamide
1-{2-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
methyl 2-{1-[(2-methyl-5-sulfamoylphenyl)carbamoyl]pyrrolidin-3-yl}acetate
(1R,7S)-3-(2-ethylbutyl)-6-(5-hydroxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-[(4-fluorophenyl)methyl]-1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane