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N-cyclopentyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
4-{4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl}-5-methylpyrimidin-2-amine
2-{4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl})amine
4-phenyl-1-(pyridin-3-ylmethyl)azepane
5-[1-ethyl-3-(3-methoxyphenoxymethyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-{[4-(naphthalen-1-yl)-5-(piperidin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(4-{[(cyclobutylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
(3S,4S)-4-(4-fluorophenyl)-1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-3-ol
methyl 4-({2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamido}methyl)benzoate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]methanol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(3-hydroxypropyl)amino]methyl}piperidin-2-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-3-methylbutanamide
4-{3-[2-methyl-3-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2,3-thiadiazole
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
6-methyl-5-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
[4-(2-aminopyridin-4-yl)phenyl]methanol
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]quinoline-3-carboxamide
3-{1-[2-(2H-indazol-2-yl)acetyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
1-ethyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-ethyl-1-(4-phenylbutanoyl)-1,4-diazepan-5-one
3-(2,3-dimethoxyphenyl)-6-(4-fluorophenyl)pyridazine
(3S,7S,8aS)-7-({[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-[(4-chlorophenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-{2,7-diazaspiro[4.5]decan-7-yl}-N-(3,5-dimethylphenyl)-2-oxoacetamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
2-(5-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1H-1,3-benzodiazole
N,2-dimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-indole
5-{3-oxo-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propyl}imidazolidine-2,4-dione
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-(2-chloro-6-methylphenyl)-4-(3-methoxypropyl)piperazine-1-carboxamide
(1R,3S,5S)-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(2-phenylethyl)piperidine-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
3-(4-fluorophenyl)-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperazin-2-one
4-[6-(2-fluoro-5-methylphenyl)pyridine-3-carbonyl]morpholine
3-(3-methoxyphenoxymethyl)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
dimethyl({4-methyl-5-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
3-benzoyl-N-(2,4,6-trimethylpyridin-3-yl)piperidine-1-carboxamide
1,3-dimethyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-1H-pyrazolo[3,4-d]pyrimidine
1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-3-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)urea
4-chloro-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,8aR)-1-butyl-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(2-oxopyrrolidin-1-yl)acetamide
1-(1'-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
9-[(2-ethoxyphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one