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4-(1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)pyridine
2-(3-methanesulfonylpropanoyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
8-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}thiolan-3-amine
1-(2-fluorophenyl)-N,2,2-trimethyl-N-(pyrimidin-4-ylmethyl)cyclopropane-1-carboxamide
N-{1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
N-cycloheptyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-fluoropyridine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-phenylbutanamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
4-(2H-1,3-benzodioxol-5-yloxy)-1-(6-methylpyridin-2-yl)piperidine-4-carboxylic acid
5-methoxy-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-pyran-4-one
2-(dimethylamino)-2-(4-methylphenyl)-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}acetamide
(1S,5R)-6-methyl-3-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-methylpyrimidin-2-amine
N4-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidin-4-yl}propanamide
1-(2-{1-ethyl-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-6-methylpyrimidin-2-amine
1-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
5-(benzenesulfonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-cyclopropanecarbonyl-4-[3-(phenoxymethyl)piperidine-1-carbonyl]piperidine
N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}quinoxaline-5-carboxamide
8-[3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-(1H-indol-2-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(dimethylamino)-2-(4-methylphenyl)acetamido]cyclopentane-1-carboxamide
1-methyl-2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
3-chloro-N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)methyl]-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[(4-chlorophenyl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
8-methoxy-2-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}quinoline
2-{1-cyclopentyl-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-methyl-2-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-({[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)-6-methoxyphenol
N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[4-(furan-2-yl)phenyl]-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
(2S,4R)-4-hydroxy-1-{3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidine-2-carboxylic acid
2-butyl-4-methyl-N-(4-methyl-3-propanamidophenyl)-3-oxopiperazine-1-carboxamide
N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
2-(adamantan-1-ylsulfanyl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
methyl 4-({2-[(2-fluorophenyl)methyl]-1,3-benzoxazol-6-yl}formamido)butanoate
1-(3-methoxyphenyl)-4-[3-(3-methoxyphenyl)propanoyl]piperazin-2-one
1-(5-amino-1H-pyrazole-3-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-benzyl-N-[2-(dimethylamino)ethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-(3-{[(1,3-benzoxazol-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
ethyl 6-[2-(methoxycarbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyridine-3-carboxylate