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N-cyclobutyl-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N,2-dimethyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
1-ethyl-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-3-methylpiperidine-3-carboxamide
1-methyl-5-[2-(oxan-2-ylmethoxy)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1S,5R)-6-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-{3-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidin-3-amine
3-propyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidine-3-carboxylic acid
3,6,7-trimethyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1-benzofuran-2-carboxamide
5-[(2S)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
2-(1H-imidazol-1-yl)-1-{2-[5-(1,4-oxazepane-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}ethan-1-one
(1S,5R)-3-[(3-ethoxy-4-methoxyphenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(1R,9aR)-1-({[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-[2-(1H-imidazol-4-yl)ethyl]-2,6-dimethylquinoline-3-carboxamide
5,6-dimethyl-2-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
2-{3-[2-(methylsulfanyl)ethyl]-5-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-{4-[2-(1-propylpiperidin-4-yl)acetyl]piperazin-1-yl}benzonitrile
4-[(3-methoxypropyl)amino]-5-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2-methoxyphenyl)methyl]methylamine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
2-{[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}morpholine
5-chloro-6-oxo-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,6-dihydropyridine-3-carboxamide
5-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-methyl-5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]quinoline
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-amino-5-methylpyrimidin-2-yl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylic acid
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[(2,4,5-trimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-methyl-N-[1-(thiophen-2-yl)propyl]pyrimidine-5-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-ol
N-butyl-4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidine-1-carboxamide
2-fluoro-4-{[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}phenol
4-{2-[methyl(phenyl)amino]acetyl}-1-(4-methylphenyl)piperazin-2-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-(2,3-difluorophenoxymethyl)-N-[(2-methoxyphenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
(1R,5S,6S)-6-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
2-{2-[(3,4-dimethylpiperazin-1-yl)methyl]-4-(4-fluorophenyl)phenoxy}acetic acid
2-acetyl-8-[(2,5-dichlorophenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(3-chloro-4-methoxyphenyl)-4-(1,4-oxazepane-4-carbonyl)pyrrolidin-2-one
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-{2-[6-(benzyloxy)pyridin-3-yl]pyrimidin-4-yl}piperidin-4-ol
N,2-dimethyl-7-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
3-fluoro-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
1-methyl-8-(3-methylpyrazin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
({2-[(3-fluorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)[(3,4,5-trimethoxyphenyl)methyl]amine
N-[3-(1H-imidazol-1-yl)propyl]-1,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-[(2-fluorophenyl)formamido]-N-[2-(1H-1,2,4-triazol-1-yl)propyl]propanamide
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide