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5,7-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[(1R,2R)-2-hydroxycyclohexyl]-1,3-oxazole-4-carboxamide
1'-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(benzyloxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(propan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]piperidine-4-carboxamide
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-[4-(1H-indol-2-yl)phenyl]pyrrolidine-1-carboxamide
3-chloro-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
2-[(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]-2-methylpropanamide
(3R,4R)-N-benzyl-4-cyclopropyl-4-hydroxy-N,3-dimethylpiperidine-1-sulfonamide
1-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-ethylurea
N-{2-[(3-{[(2,5-dimethoxyphenyl)methyl]amino}-5-(dimethylsulfamoyl)phenyl)formamido]ethyl}acetamide
N-(2-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]amino}ethyl)acetamide
3-hexyl-8-(2-methyl-1,3-thiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-cyclopropanecarbonyl-2-[(3,4-dimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(3-hydroxyphenyl)methyl]piperidine-4-carboxylic acid
[(3R,4R)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3aR,6aR)-2-cyclopentyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-{2-hydroxy-3-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]propyl}piperidin-4-ol
4-(furan-2-yl)-2-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-5-(propan-2-yl)-1H-pyrazol-1-yl)pyrimidine
3-(2-chlorophenoxy)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}azetidine
(1S,5R)-3-(2,2-diphenylethyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(3-cyclopentylpropanoyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-cyclobutyl-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole
N'1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N'1-methylcyclopropane-1,1-dicarboxamide
N-(1,2-oxazol-3-ylmethyl)-4-(piperazine-1-carbonyl)benzene-1-sulfonamide
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
1-[4-(methoxymethyl)piperidin-1-yl]-3-(2-methylphenyl)-3-phenylpropan-1-one
[(8-chloroquinolin-2-yl)methyl](methyl)(oxan-4-ylmethyl)amine
(4-{[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]amino}quinazolin-2-yl)methanol
6-fluoro-4-(pyridin-2-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-(1H-1,2,3-triazol-1-yl)acetamide
2-(4-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
N-[(5-methylpyrazin-2-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(1R,5S)-3-({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
4-(furan-2-ylmethyl)-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-[3-(dimethylsulfamoyl)propyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(1H-1,2,3-benzotriazol-5-yl)-3-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carboxamide
(1R,5R)-6-{[3-(furan-2-yl)phenyl]methyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
2-(4-methylphenyl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
5-(2-fluorophenyl)-N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[(2,5-dichlorophenyl)formamido]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
ethyl 4-(2-phenoxyethyl)-1-(quinolin-8-ylmethyl)piperidine-4-carboxylate
(1S,5R)-6-(2-methoxyethyl)-3-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine