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2-[5-(3,4-difluorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
(1S,5R)-6-{3-[(3-fluorophenyl)methoxy]benzoyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-(1H-imidazol-2-ylmethyl)-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrrolidin-3-ol
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2,5-dimethyl-1,3-oxazole
(2S)-2-amino-3-hydroxy-1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
1-[4-(cyclopropylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
5-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridin-2-amine
5-(3-methoxyphenyl)-3-(4-methyl-3-phenylpiperazin-1-yl)-1,2,4-triazine
2-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}-1-phenylethan-1-ol
4-{[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyridine
3-{[3-cyclopropyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2,5-oxadiazole
1-[3-(6-hydroxy-1,4-oxazepan-4-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
3-{1-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]piperidin-3-yl}propan-1-ol
6-methyl-2-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
(1R,2S)-N-butyl-2-{3-oxo-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepine-6-carbonyl}cyclohexane-1-carboxamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
3-{1-[2-(naphthalen-2-yloxy)propanoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
2,6-dimethyl-4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenyl acetate
1-(2-cyclohexylethyl)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-({[4-(1H-imidazol-1-yl)phenyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methylpiperidin-3-ol
1-{4-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]pyrimidin-2-yl}piperidine-4-carboxamide
2-[4-(dimethylsulfamoyl)morpholin-3-yl]-N-(2-phenoxyethyl)acetamide
2-(2,3-dimethoxy-5-methylphenyl)-N,N-dimethylbenzamide
8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-N-(propan-2-yl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
6-{6-hydroxy-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-1-yl}pyrazine-2-carboxamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(morpholine-4-sulfonyl)benzamide
2-(morpholin-3-yl)-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}acetamide
1-{2-oxo-2-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethyl}piperidin-2-one
(1R,9aR)-1-{[(2-methylbut-3-yn-2-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
6-(2,2-diethylmorpholin-4-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
3-{[cyclohexyl(methyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
[(3R,4R)-1-(3,5-dichlorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(4aS,8aR)-6-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2-methylphenol
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]urea
N-{1-oxaspiro[4.4]nonan-3-yl}-4-(propylsulfamoyl)benzamide
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)methylamine
5-(5-methylfuran-2-yl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1,2,4-triazin-3-amine
N-({1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-3-yl}methyl)-5-methoxyfuran-2-carboxamide
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-[(3-fluorophenyl)methyl]piperazine
(2R,3R,6R)-5-(oxane-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carboxamide