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methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl][(3-phenyl-1H-pyrazol-4-yl)methyl]amine
N-methyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(thiophen-3-ylmethyl)acetamide
3-(4-hydroxyphenyl)-N-methyl-N-(prop-2-en-1-yl)benzamide
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-1-benzofuran-2-carboxamide
N-[(3R,4R)-1-[2-(4-ethylpiperazin-1-yl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(4aR,7aS)-1-benzyl-4-(4-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
5-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)-2-(methylsulfanyl)pyrimidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-2-(pyridin-2-yl)acetamide
4-({4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]urea
2-(dimethylamino)-1-[1-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-(2-methoxyphenyl)-3-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(trifluoromethyl)pyridine
3-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
3-cyclopentyl-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
2-(methoxymethyl)-6-methyl-3-[4-(2-methylphenyl)piperazine-1-carbonyl]-1-(naphthalen-1-ylmethyl)-1,4-dihydropyridin-4-one
(2S,4S)-4-amino-N-[2-(3-methoxyphenyl)ethyl]-1-methylpyrrolidine-2-carboxamide
(2S,4R)-4-amino-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-N-methylpyrrolidine-2-carboxamide
2-(1H-indol-5-yl)-1H-1,3-benzodiazole-5-carbonitrile
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}methanesulfonamide
2-{5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-cyclopentyl-1H-1,2,4-triazol-1-yl}acetic acid
N-({1-[(3-ethenylphenyl)methyl]piperidin-3-yl}methyl)acetamide
2-(4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
1-(5-ethylthiophene-3-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(1S,5R)-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(1,2-oxazinan-2-yl)propanamide
(2R)-N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]pyrrolidine-2-carboxamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
(3S,5R,9R)-11-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N5-(3-methylbutyl)-N3-(1-methylpiperidin-4-yl)-1-(2-methylpropyl)-4-oxo-N3-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]urea
9-(2-methoxybutanoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(5-ethylpyridin-2-yl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
3-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
(2S,3S)-2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-3-methylpentanamide
1-[2-(1-ethyl-1H-pyrazol-4-yl)-3,6-dimethylquinoline-4-carbonyl]piperidine-3-carbonitrile
(3S,4R)-1-(2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
(3aS,6aS)-5-[(5-methylthiophen-2-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-4-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
(2S,4S)-4-amino-N-ethyl-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]pyrrolidine-2-carboxamide
2-(furan-2-yl)-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)azepane
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2,4-dimethylphenoxy)ethyl]methylamine
1-(3-phenylpropanoyl)-4-propyl-1,4-diazepan-5-one
N-ethyl-N-{1-[3-(2-methyl-1H-indol-1-yl)propanoyl]pyrrolidin-3-yl}acetamide
2-(4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
5-(2-fluorophenyl)-N-[(2S)-oxolan-2-ylmethyl]pyrazolo[1,5-a]pyrimidin-7-amine