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1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one
3-(4-chlorophenyl)-N-methyl-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
4-(pyridin-2-ylmethyl)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
3-chloro-4-({1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]benzene-1-sulfonamide
N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
1,4-dimethyl-2-({1-[(3-methylphenyl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl}methyl)piperazine
1-phenyl-4-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepane
2-(cyclopropylmethyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]morpholine
[(3R,4R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
3-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]propan-1-ol
4-cyclobutyl-N,6-dimethyl-N-[(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine
3-[3-(propan-2-yloxy)benzoyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-(2-{[7-acetyl-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)acetamide
2-{4-[(4-methylnaphthalen-1-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetic acid
5-(dimethylamino)-2-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}ethane-1-sulfonamide
N-[2-(azepan-1-yl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(propan-2-yl)acetamide
2-(4-fluorophenyl)-N-[2-(pyridin-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-[(1-benzylpiperidin-4-yl)amino]-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
methyl (2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-(4-methoxybenzamido)pyrrolidine-2-carboxylate
N,1,3-trimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(3-acetyl-1H-pyrazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
N-methyl-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
4-cyano-N-(5-acetamido-2-fluorophenyl)piperidine-1-carboxamide
4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-one
(2S,4R)-N-ethyl-4-(furan-2-amido)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxamide
N-[2-(3-methoxyphenyl)-1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-(4-methylphenyl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
N-[(3R,4R)-3-hydroxy-1-(quinoxalin-2-yl)piperidin-4-yl]pyrazine-2-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1-(4-methylphenyl)cyclopropane-1-carboxamide
5-chloro-N-(3-hydroxy-3-methylbutyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
3-({[2-(cyclopentyloxy)phenyl]methyl}(methyl)amino)-N-methylbutanamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
8-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-(2H-1,3-benzodioxol-5-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2,4-triazin-3-amine
N-[3-(3-methoxyphenyl)phenyl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine-4-carboxamide
N-[2-(3-methoxyphenyl)-1-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
5-{2-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(4-phenylphenyl)acetamide
1-(1H-1,3-benzodiazole-2-carbonyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
3-(2-fluorophenyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-phenylpropanamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-(dimethylamino)acetamide