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2-methoxy-5-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}benzoic acid
(3aR,5R,6S,7aS)-2-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
5-(2-fluorophenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(3-chloro-4-hydroxyphenyl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]ethan-1-one
3-cyclopropyl-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
2,2,3,3-tetramethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]cyclopropane-1-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyrimidine-2,4-diamine
N,N-dimethyl-2-(pyridin-4-yl)-7-(pyridine-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-methyl-4-(morpholin-4-yl)benzamide
1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-5-(pyrrolidin-1-ylmethyl)-1H-imidazole
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(pyridin-3-yloxy)ethyl]benzamide
[3-propyl-1-(4,4,4-trifluorobutyl)piperidin-3-yl]methanol
ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-(cyclopentylmethyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-phenylpiperidine-4-carbonitrile
methyl 5-{[(2-methoxyphenyl)methyl]amino}-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
2-(2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenoxy)acetic acid
2-(4-fluorophenyl)-N-(1-methoxybutan-2-yl)imidazo[1,2-a]pyridine-6-carboxamide
3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-methyl-3-(2-methylpropyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-oxazole-5-carboxamide
3-phenyl-8-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
2-amino-4-(5-methylfuran-2-yl)-6-[4-(morpholin-4-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
1-cyclohexyl-3-(cyclopropylmethyl)-N-[2-(dimethylamino)ethyl]-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-fluoroethyl)acetamide
(4aS,7aR)-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-ethyl-2-methyl-N-[1-(pyridin-4-yl)propyl]pyrimidin-4-amine
1-(2,2-dimethyloxan-4-yl)-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
3-(2-fluorophenoxymethyl)-1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-methyl-6-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-4H-pyran-4-one
(3aS,6aS)-5-(3,6-dimethylpyrazin-2-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(3-methylbutanoyl)-4-[(6-methylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-cyclopropyl-5-(morpholin-4-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(methylsulfanyl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-[(4-fluorophenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(2-methylphenyl)sulfanyl]ethan-1-one
N-cyclopropyl-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
3-[2-(piperazin-1-yl)ethyl]-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[4-(morpholin-4-yl)butyl]amine
2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one