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N-[2-(pyrrolidin-1-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
5-(2-chlorophenyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}furan-2-carboxamide
1-({1-[(2-chloro-6-fluorophenyl)methyl]-3-cyclopentyl-1H-1,2,4-triazol-5-yl}methyl)pyrrolidin-2-one
N,N-bis(1,3-oxazol-4-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-methyl-4-(4-methylquinolin-2-yl)piperazine-2-carboxylic acid
N-[(4-hydroxy-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}azepan-4-yl)methyl]piperidine-1-carboxamide
2-(2-methoxyethyl)-8-[(1-methyl-1H-indol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(1H-imidazol-1-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]acetamide
2-(3-chloro-4-fluorophenyl)-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}acetic acid
2-(3-fluorophenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopentyl-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-N-(pyridin-3-yl)propanamide
1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepan-6-ol
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-phenylethyl)acetamide
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-[3-(propan-2-yloxy)propyl]propanamide
methyl 1-({4-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
1-(isoquinolin-1-yl)-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
4-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-ethyl-5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
2,6,8-trimethyl-4-[3-(piperidin-1-yl)azetidine-1-carbonyl]quinoline
2-(3-methoxypropyl)-9-(1H-1,2,4-triazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1-methylpiperidine
1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-4-(pyridin-4-yl)piperazine
3-({[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)propane-1,2-diol
N-cyclopropyl-15-methyl-13-oxo-9-phenyl-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
4-{1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazine-1-carbaldehyde
(2S,4S,5R)-2-ethyl-4-(3-hydroxyazetidine-1-carbonyl)-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
6-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}quinoxaline
2-(2,5-dimethoxyphenyl)-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
9-(4-methoxy-3-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-2-(piperidin-1-yl)pyrimidine
N-{[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-(3,3,3-trifluoropropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1H-imidazol-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylbenzamide
3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
N-[3-(azepan-1-yl)propyl]-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
N-phenyl-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
1-{2-hydroxy-3-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}piperidin-4-ol
3-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-phenyl-1,2-oxazole
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
1-cyclopentyl-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-2-one
3-[({1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide