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4-phenyl-3-({1-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[3-(3,4-difluorophenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]propan-2-yl}acetamide
[(4-ethylphenyl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-[1-(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
(1-methyl-5-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
3-[3-(2-cyclopentylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-(1H-1,3-benzodiazol-1-yl)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}propan-1-one
(2S,4S)-4-amino-N-(1-carbamoylcyclopentyl)-1-methylpyrrolidine-2-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(2-benzyl-5-oxopyrrolidin-2-yl)propanamide
(3S,4R)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[(3S,4R)-1-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N3-butyl-1-(furan-2-ylmethyl)-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-1λ6-thiomorpholine-1,1-dione
3-ethyl-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-3-carboxylic acid
(3R,5R)-1-[(3,4-dimethoxyphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
(3R,4R)-1-(4-methoxybenzoyl)-4-[(3-phenylpropyl)amino]pyrrolidin-3-ol
1-(azocan-1-yl)-3-[5-methoxy-2-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
1-(3-chloro-2-fluorophenyl)-3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]urea
4-ethyl-1-methyl-3-{[1-(pyrazine-2-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-phenyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)-N-phenylpropanamide
(1S,5R)-3-(2-methyl-6-propylpyrimidin-4-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2-methoxyphenyl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
5-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(pyridin-3-yl)pyrimidine
1-(2-fluorophenyl)-4-(1-propylpiperidin-4-yl)piperazine
N-benzyl-2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]acetamide
N,1,3,7-tetramethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
methyl (2S,4S)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
4-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)pyridine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(methylamino)pyridine-4-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-[(5-ethylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(3-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]acetamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylpentan-1-one
4-[1-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)piperidin-3-yl]benzoic acid
2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridin-3-ol
7-oxo-5-(5-propyl-1,2-oxazol-3-yl)-2-(pyrrolidin-1-yl)-4H,7H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile
(2S)-2-amino-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-phenylethan-1-one
5-methyl-1-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1-(cyclopropylmethyl)-4-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]piperazin-2-yl]ethan-1-ol
(2S,4S)-4-amino-1-[2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1-(3-fluorophenyl)-3-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
4-methyl-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)-1,4-diazepane-1-carboxamide
4-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-2,2,6,6-tetramethylpiperidine
2-(2-hydroxyethyl)-6-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-(4-methoxyphenyl)-4-{[2-(methylsulfanyl)phenyl]methyl}piperazin-2-one