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methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]heptanoic acid
methyl 6-[(diethylamino)methyl]-3-(2,3-dimethylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
3-(5-acetyl-2-ethoxyphenyl)-1-(3-hydroxy-3-phenylpropyl)-1-methylurea
5-methanesulfonyl-4-(piperidin-3-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
N-(1,4-dioxan-2-ylmethyl)-6-ethyl-N-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methyl-2-[(4-methylphenyl)amino]propanamide
1-{3-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]propyl}-2,3-dihydro-1H-imidazol-2-one
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-4-methylphenol
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2,6-dimethoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
5-[1-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
1-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)-4-phenylpiperazine
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-5-methyl-1,3-oxazole
2-cyclobutyl-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-4-(morpholin-4-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-[4-(quinolin-2-yl)-1H-1,2,3-triazol-1-yl]propane-1,2-diol
2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
{4-[(4-propoxyphenyl)methyl]morpholin-2-yl}methanamine
2-{2-[(1-phenoxypropan-2-yl)amino]ethyl}-3,4-dihydroquinazolin-4-one
6-(phenoxymethyl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(methoxymethyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}cyclobutane-1-carboxamide
N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
1-cyclopentanecarbonyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
4-(3-methylpiperidin-1-yl)-3-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetamido]benzamide
7-(1,2-oxazole-3-carbonyl)-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
9-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-methoxy-4-phenyl-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
2-amino-3-ethyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(4-fluorophenyl)ethyl]-1-methyl-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
(3aS,6aS)-2-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
5-ethyl-1'-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-benzyl-3-[1-(pyrimidin-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-5-[1-(3-hydroxy-4-methoxybenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
3-[(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)methyl]phenol
2-ethyl-9-(1-phenylcyclopropanecarbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[2-(dimethylamino)ethyl]amino}-N,N,5-trimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-N-[2-(oxan-4-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})(quinolin-5-ylmethyl)amine
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
methyl 2-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-5-methoxy-N-(oxolan-2-ylmethyl)furan-2-carboxamide
2-methoxy-N-[(3R,5S)-1-(3-methoxypropyl)-5-(methylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-{4-[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]piperidin-1-yl}ethan-1-one
1-[6-(3,4-dimethylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]azepane
2-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)pyridine-3-carboxylic acid