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2-[4-(acetamidomethyl)piperidin-1-yl]pyridine-4-carboxamide
2-{[benzyl(methyl)amino]methyl}-4-phenylphenol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N'-(2,5-dimethoxyphenyl)propanediamide
2-[1-(2-methoxyethyl)piperidin-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(4-methoxyphenyl)-N-[(6-methylpyridin-2-yl)methyl]-3-phenylpropanamide
2-[1-(3,4,5-trimethoxyphenyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-N-{2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]ethyl}pyridin-4-amine
2-(3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}phenoxymethyl)pyridine
4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}morpholine-2-carboxylic acid
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentan-1-one
(3S,4S)-1-(2-fluorobenzoyl)-4-(naphthalen-2-yl)piperidin-3-ol
5-[(benzyloxy)methyl]-3-methyl-1-phenyl-1H-1,2,4-triazole
N-methyl-2-(2-phenyl-1H-imidazol-1-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]acetamide
2-amino-3-ethyl-N-[2-(piperidin-1-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-1-(pyrimidin-2-yl)piperidine-4-carboxamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
N-[2-(2-fluorophenoxy)pyridin-3-yl]-2-methyl-1,4-oxazepane-4-carboxamide
1-benzyl-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-2-one
4-(5-ethyl-1,3-oxazole-4-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
6-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
4-hydroxy-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
2-methyl-3-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}-2,8-diazaspiro[4.5]decane
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
1-(4-chloro-2-methoxybenzoyl)-2-(3-methoxypropyl)piperidine
1-({[1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
N-(3,5-dimethylphenyl)-N'-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanediamide
1-[1-(4-hydroxybenzoyl)piperidin-3-yl]-2-phenylethan-1-one
4-(piperidine-1-carbonyl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-4-yl}methanesulfonamide
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-1,2,3,6-tetrahydropyridine
2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-6-(4H-1,2,4-triazol-4-yl)pyridine
N-(3,5-dimethoxyphenyl)-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]propanamide
6-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-N-ethyl-N-methylpyridine-3-carboxamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(2-fluoro-3-methoxyphenyl)oxan-4-yl]acetamide
(3R,5S)-1-(naphthalen-2-ylmethyl)-N-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-(3-phenylpropyl)-8-[3-(1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aR)-6-[(2,3-dichlorophenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl){2-[(4-methylphenyl)sulfanyl]ethyl}amine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2,1-benzoxazole-3-carboxamide
3-(4-methoxyphenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-phenylpropanamide
4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-[(3S,4R)-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}-4-propylpyrrolidin-3-yl]acetamide
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-(propan-2-yl)propanamide
4-(5-ethylpyridin-2-yl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{[(3S,4S)-1-(2,6-dimethoxypyridine-3-carbonyl)-3-hydroxypiperidin-4-yl]methyl}-3,3-dimethylurea
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-(1H-pyrazol-1-yl)butan-1-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-2-oxo-N-(prop-2-en-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
2-{4-[(2-methoxyphenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
N-tert-butyl-1-(3-methylbutyl)-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide