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N-[(3-fluoro-4-methylphenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}piperidine-3-carboxamide
5-benzoyl-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-cyclohexyl-N-[(2,6-difluoro-3-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-methyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-5-phenylthiophene-2-carboxamide
3-chloro-N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2-methyl-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-propylacetamide
(3S,4R)-4-(4-fluorophenyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidine-3-carboxylic acid
N-[2-(2-methyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethyl]-N-(4-methylphenyl)methanesulfonamide
(4aS,7aR)-1-(2-hydroxypyridine-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[4-(3-fluorophenyl)benzoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)ethane-1-sulfonamide
8-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
4-(4-{[(2-hydroxypropyl)(methyl)amino]methyl}phenyl)-2-methylbutan-2-ol
N-[2-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)ethyl]acetamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-(2-chlorophenyl)ethyl}-N-methylfuran-2-carboxamide
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
1-[2-(4-methoxyphenyl)phenyl]-3-[2-(propane-2-sulfonyl)ethyl]urea
2-methyl-4-(4-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
2-benzyl-9-[(3R)-3-hydroxy-3-phenylpropyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-(2,6-dimethylphenyl)-3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)benzamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-(3-fluorophenyl)-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)benzamide
N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]benzamide
N-[(3-methoxyphenyl)methyl]-3-{1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}propanamide
N-({8-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
8-[(2E)-3-phenylprop-2-enoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(cyclohex-1-en-1-yl)-4-methoxy-N-methylbenzamide
4-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
6-ethyl-2-[2-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}urea
(3aR,6aR)-2-cyclopentyl-N-[3-(morpholin-4-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]benzamide
(3R,4R)-4-ethyl-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine-3,4-diol
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(4-phenyloxan-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N3-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
methyl (1R,3S,3aR,6aS)-3-[3-(furan-2-yl)phenyl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amine
3-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
5-{2-[2-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-N-(trimethyl-1H-pyrazol-4-yl)benzamide
4-chloro-5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)-1,3-thiazole
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazine
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-methyl-2-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenol