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N-benzyl-2-[(dimethylamino)methyl]-N-(3-hydroxy-2-methylpropyl)-1,3-thiazole-4-carboxamide
1-cyclopropanecarbonyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)piperidine-4-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-ol
N-cyclopropyl-N-[(4-methoxyphenyl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-cyclopropyl-4-methoxy-2-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-methyl-7-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-2H-chromen-2-one
N,1-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrrole-2-carboxamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]thiophene-3-sulfonamide
2-[2-(propan-2-yloxy)phenyl]-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
2,6-dimethyl-N-[(1R,2S)-2-phenylcyclopropyl]pyridine-4-carboxamide
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-methylpentan-1-one
1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]urea
2-(azocan-1-yl)-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-N-[(1-methylpyrrolidin-3-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
2-{4-[4-chloro-3-(1H-pyrrol-1-yl)benzoyl]morpholin-3-yl}acetic acid
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(1H-pyrazol-1-yl)benzamide
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
5-[2-(1H-imidazol-5-yl)-1-(1H-pyrrol-1-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-oxo-2H-chromene-3-carboxamide
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
5-{1-[(3-cyanophenyl)methyl]pyrrolidin-2-yl}-N-cyclopentylthiophene-2-carboxamide
N-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
6-{4-[(3,5-dichloropyridin-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
2-{[5-(ethoxymethyl)-4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-{[4-(3-methylphenyl)phenyl]methyl}piperazin-2-one
1-(3-fluorophenyl)-5-(1-methoxy-2-methylpropan-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-methoxy-5-methylbenzene-1-sulfonamide
N-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}methanesulfonamide
(1R,7S)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}-3,5-dimethyl-1H-pyrazole
3-{1-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
2-(2-hydroxyethyl)-9-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(azepane-1-carbonyl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
6-methyl-N4-[(6-methylquinolin-5-yl)methyl]pyrimidine-2,4-diamine
3-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]benzonitrile
(4aR,7aS)-1-cyclobutanecarbonyl-4-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-methanesulfonamidopropanamido)-N-methyl-N-phenylbenzamide
1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
3-(4-fluorophenoxymethyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
methyl 2-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methylacetamido]acetate
(2S,4S)-4-(3-cyanobenzamido)-N-ethyl-1-(furan-2-ylmethyl)pyrrolidine-2-carboxamide