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(3S)-1-ethyl-3-methyl-4-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
1-({5-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(oxan-2-ylmethyl)pyrimidin-2-amine
(3R)-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-[methyl(phenyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
1-(1-hydroxynaphthalene-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-1,3-thiazole-4-carboxamide
3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(3-fluorophenyl)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-benzyl-N3-butyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
4-(1-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-methylpropan-2-yl)morpholine
N-[2-(2-fluorophenyl)-1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
3-{4-[1-(2-methoxyphenyl)-3-phenylprop-2-yn-1-yl]piperazin-1-yl}propanamide
N-(2-methyl-1-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-1-oxopropan-2-yl)thiophene-2-carboxamide
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-1,3-oxazole-5-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
1-(2-aminopyridine-4-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
3-{[4-(3-chlorophenyl)-5-{[methyl(thiophen-3-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepan-5-one
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](ethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
2-(5-acetamido-1H-1,2,4-triazol-3-yl)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-(2,2-dimethylpropanoyl)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
1-[2-hydroxy-3-(2-methoxy-4-{[(3-phenylpropyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
6-[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2-amino-4-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}quinazoline-6-carboxylic acid
3-(4-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)propanamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(furan-2-ylformamido)methyl]benzoate
5-({[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl](propan-2-yl)amino}methyl)pyrrolidin-2-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-4-yl)propan-1-one
8-[(3-hydroxy-4-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
8-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N'-cyclopentyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)ethanediamide
3-fluoro-N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(azepan-1-yl)-3-[3-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-amido)cyclopentane-1-carboxylic acid
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-(pyridin-3-ylmethyl)piperidin-4-amine
N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-[6-(methoxymethyl)pyrimidin-4-yl]-7-methyl-1H-indole
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
N-[(3R,4S)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(pyridin-2-yl)pyrrolidin-3-yl]acetamide
2-amino-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
4-[5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidin-2-yl]morpholine
(2R,3R)-1'-(2,1,3-benzoxadiazol-4-ylmethyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol