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2-(adamantan-1-yl)-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
1-ethyl-N,3-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propan-1-one
methyl 2-{8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
8-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-fluorophenyl)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperazin-2-one
N,5-dimethyl-2-(2-methylpropanamido)-N-(1H-pyrazol-5-ylmethyl)benzamide
(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-amino-N-methyl-1-[2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetyl]pyrrolidine-2-carboxamide
2-[4-({[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl](methyl)amino}methyl)piperidin-1-yl]ethan-1-ol
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-hydroxyphenyl)ethan-1-one
6-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-7-methyl-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
1-[(4aR,8aR)-4a-hydroxy-7-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
4-ethyl-N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}carbamoyl)amino]-N,N,3-trimethylbenzamide
8-[3-(2-methoxyphenyl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(2S,4R)-4-{[(2,4-difluorophenyl)methyl]amino}-N-methyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
1-[2-(dimethylamino)ethyl]-N-(naphthalen-1-ylmethyl)-5-oxopyrrolidine-3-carboxamide
(2S)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2,3-dihydro-1H-indole-2-carboxamide
2-(3-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}phenoxy)acetamide
N-methyl-2-(1H-pyrazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
4-(2,3-difluoro-4-methoxybenzoyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
6-[4-(2,6-dimethylpyridine-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
5-[({2-[(3-chlorophenyl)carbamoyl]ethyl}amino)methyl]-N-methylfuran-2-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2,8-dimethylquinoline-4-carboxamide
1-[2-(azepan-1-yl)ethyl]-3-[4-(difluoromethoxy)phenyl]-1-methylurea
N,6-dimethyl-2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
6-{4-[(dimethylamino)methyl]phenyl}-N-(propan-2-yl)pyrimidin-4-amine
1-ethyl-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3S,4R)-1-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2,4-dimethoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1-methyl-3-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-[(2,3-difluoro-4-methylphenyl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
N-methyl-2-(morpholin-3-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(2S,4S)-1-cyclopentyl-N-ethyl-4-[2-(4-methoxyphenyl)acetamido]pyrrolidine-2-carboxamide
2-(methylamino)-N-[2-(2-phenoxyethoxy)phenyl]acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
3-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-6-methyl-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-2-one
[(2-butyl-1H-imidazol-4-yl)methyl]({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-{9-[(3-methoxyphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-ethyl-3-[1-(propan-2-yl)-5-[(propan-2-yl)sulfamoyl]-1H-1,3-benzodiazol-2-yl]propanamide
5-fluoro-N4,N4-dimethyl-N2-[(3-methyl-1-benzofuran-2-yl)methyl]pyrimidine-2,4-diamine
5-benzyl-1-(4-methylphenyl)-4-(pyrazine-2-carbonyl)piperazin-2-one
1-(4-chlorophenyl)-N-({1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide