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6-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
3-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
4-chloro-2,5-dimethyl-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
3-ethyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1H-indole-2-carboxamide
2-[2-(3-methoxyphenyl)azetidine-1-carbonyl]pyrazine
(1r,4r)-4-{[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]methyl}cyclohexane-1-carboxamide
5-[(2-benzylmorpholin-4-yl)methyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)acetic acid
4-[(1R,2S)-2-propylcyclopropanecarbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methanol
5-methoxy-N-(2-methoxyethyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
2-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)-N-cyclopentylpropanamide
(4aS,7aR)-1-(4-ethylbenzoyl)-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[4-(hydroxymethyl)benzoyl]pyrrolidin-3-yl}propan-2-ol
4-ethyl-2-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-thiazole-5-carboxamide
5-benzyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
4-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
2-[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
2-(2,2-dimethylcyclopropanecarbonyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-ethyl-3-({1-[(2-methoxypyridin-3-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-propyl-3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-butanoyl-4-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
6-(aminomethyl)-2-[4-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-(4-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)propanoic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
8-chloro-4-[4-(cyclobutylmethyl)piperazine-1-carbonyl]-2-methylquinoline
2-chloro-5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}amino)-N-(propan-2-yl)benzamide
(1R,2R)-N,N-diethyl-2-(4H-1,2,4-triazol-4-yl)cyclohexan-1-amine
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
5-[4-(diphenylmethyl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline
2-[(3-methoxyphenyl)methyl]-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(4-methylmorpholin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
2-[(1S,5R)-6-[(3,5-dimethyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
N-[2-(4-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenoxy)ethyl]acetamide
N-ethyl-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(oxolan-2-ylmethyl)acetamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(3-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(4aR,8aR)-2-[(3-chloro-2-fluorophenyl)methyl]-7-cyclobutanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
3-(1H-imidazol-2-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
8-(oxan-3-yl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
diethyl[(3-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)methyl]amine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
dimethyl(3-{2-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-methyl-4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine