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1-(4-methylphenyl)-4-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperazin-2-one
2-[(2,3-dimethyl-1H-indol-7-yl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
1-(2-chlorophenyl)-4-(2-hydroxy-4-methoxybenzoyl)-5-methylpiperazin-2-one
5-(1-aminoethyl)-N-cyclohexyl-N,4-dimethylpyrimidin-2-amine
4-({4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
4-{3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzoyl}thiomorpholine
1-{3-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]propyl}piperidine-3-carboxamide
N-{1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
2-{4-[2-methyl-3-(1H-pyrazol-1-yl)propyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
2-(2-chloro-6-fluorophenyl)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}ethan-1-one
1-ethyl-4-[({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]pyrrolidin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}acetamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
(3S,4S)-4-({[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amino}methyl)piperidin-3-ol
N-[4-(furan-2-ylmethoxy)phenyl]-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
4-(4-methylphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(pyridin-4-yl)pyrimidin-2-amine
3,5-dimethyl-4-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2-oxazole
5-methoxy-2-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]phenol
N,N-dimethyl-2-[({thieno[3,2-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[2-(furan-2-yl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-(2,5-dimethylphenyl)-6,8-dioxo-2,7-diazaspiro[4.4]nonane-2-carboxamide
2-(pyridin-2-yl)-5-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-ethyl-3-(3-hydroxyquinoxalin-2-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
ethyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
6-[(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-2-carbonitrile
(4aS,8aR)-6-[6-(morpholin-4-yl)pyrimidin-4-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
3-methyl-4-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-1,2,5-oxadiazole
3-(2-hydroxyphenyl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
{1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
4-[2-(4-chlorophenyl)morpholin-4-yl]-4-oxobutanamide
methyl 3-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-1-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
8-(2-hydroxyethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(ethylamino)-N-[1-(4-fluorophenyl)ethyl]pyrimidine-5-carboxamide
N-({5-[(4-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
3-acetyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrazole-5-carboxamide
(3S,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[2-(morpholine-4-carbonyl)piperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
4-({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
8-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-{4-[(6-chloropyridin-3-yl)methyl]piperazine-1-carbonyl}-2,8-diazaspiro[4.5]decane
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)acetamide
2-(2-aminopyrimidin-4-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[(1H-imidazol-2-ylmethyl)(propan-2-yl)amino]propanamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-2-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(morpholin-3-yl)acetamide
3-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-1-[(1-hydroxycyclohexyl)methyl]urea
6-[(E)-2-phenylethenyl]pyridine-2-carbonitrile
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide